Inhibition of matrix metalloproteinase-9 by "multi-prong" surface binding groups

Chem Commun (Camb). 2005 May 28:(20):2549-51. doi: 10.1039/b501780g. Epub 2005 Mar 7.

Abstract

A novel strategy of blocking the active site accessibility of MMP-9 by "multi-prong" surface binding groups is described.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Copper / chemistry*
  • Enzyme Inhibitors / chemistry
  • Enzyme Inhibitors / pharmacology*
  • Imino Acids / chemistry*
  • Matrix Metalloproteinase 10
  • Matrix Metalloproteinase 9 / chemistry
  • Matrix Metalloproteinase Inhibitors*
  • Metalloendopeptidases / antagonists & inhibitors
  • Metalloendopeptidases / chemistry
  • Models, Molecular
  • Molecular Structure
  • Organometallic Compounds / chemistry
  • Organometallic Compounds / pharmacology*
  • Structure-Activity Relationship
  • Surface Properties

Substances

  • Enzyme Inhibitors
  • Imino Acids
  • Matrix Metalloproteinase Inhibitors
  • Organometallic Compounds
  • Copper
  • Metalloendopeptidases
  • Matrix Metalloproteinase 10
  • Matrix Metalloproteinase 9
  • iminodiacetic acid