Use of novel, non-imidazole inverse agonist radioligands to define histamine H3 receptor pharmacology

Inflamm Res. 2005 Apr:54 Suppl 1:S46-7. doi: 10.1007/s00011-004-0421-y.
No abstract available

MeSH terms

  • Animals
  • Biphenyl Compounds / chemistry
  • Biphenyl Compounds / pharmacology*
  • Cell Line
  • Histamine Agonists / chemistry
  • Histamine Agonists / pharmacology*
  • Humans
  • Imidazoles / chemistry
  • Molecular Structure
  • Piperazines / chemistry
  • Piperazines / pharmacology*
  • Radioligand Assay
  • Rats
  • Receptors, Histamine H3 / metabolism*

Substances

  • A349821
  • Biphenyl Compounds
  • Histamine Agonists
  • Imidazoles
  • N-(2-(4-(3-(4-(cyclopropylcarbonyl)phenoxy)propyl)-1-piperazinyl)-1-methyl-2-oxoethyl)-2-furamide
  • Piperazines
  • Receptors, Histamine H3
  • imidazole