In vitro activity of a monoclonal killer anti-idiotypic antibody and a synthetic killer peptide against oral isolates of Candida spp. differently susceptible to conventional antifungals

Oral Microbiol Immunol. 2005 Aug;20(4):226-32. doi: 10.1111/j.1399-302X.2005.00217.x.

Abstract

Background/aims: A monoclonal killer anti-idiotypic antibody (mAbK10) and a synthetic killer peptide, acting as internal images of a microbicidal, wide-spectrum yeast killer toxin (KT) have been recently shown to express candidacidal in vitro and an in vivo therapeutic activity against experimental mucosal and systemic candidosis models caused by a reference strain of Candida albicans (10S).

Material and methods: The in vitro candidacidal activity of mAbK10 and synthetic killer peptide was compared using a colony forming unit assay against a large number of isolates of different Candida spp., obtained from oral saliva of adult diabetic (type 1 and 2) and nondiabetic subjects from Parma (Italy) and London (UK).

Results: Both the KT-mimics exerted a strong dose-dependent candidacidal activity, probably mediated by the interaction with beta-glucan KT receptors on target yeast cells, against all the tested strains, regardless of their species and pattern of resistance to conventional antifungal agents.

Conclusions: These observations open new perspectives in the design and production of candidacidal compounds whose mechanism reflects that exerted in nature by killer yeasts.

MeSH terms

  • Adult
  • Animals
  • Antibodies, Anti-Idiotypic / pharmacology*
  • Antibodies, Fungal / pharmacology*
  • Antibodies, Monoclonal / pharmacology
  • Antifungal Agents / pharmacology*
  • Candida / drug effects*
  • Candida / immunology
  • Colony Count, Microbial
  • Diabetes Mellitus / immunology
  • Dose-Response Relationship, Drug
  • Drug Design
  • Humans
  • Killer Factors, Yeast
  • Microbial Sensitivity Tests
  • Mycotoxins / pharmacology*
  • Protein Engineering
  • Rats
  • Recombinant Proteins / pharmacology
  • Saliva / microbiology

Substances

  • Antibodies, Anti-Idiotypic
  • Antibodies, Fungal
  • Antibodies, Monoclonal
  • Antifungal Agents
  • Killer Factors, Yeast
  • Mycotoxins
  • Recombinant Proteins
  • killer toxin, Pichia