Effects of estrogen, raloxifene, and hormone replacement therapy on serum C-reactive protein and homocysteine levels

Maturitas. 2006 Feb 20;53(3):252-9. doi: 10.1016/j.maturitas.2005.05.006. Epub 2005 Jun 28.

Abstract

Objectives: To investigate the effects of conjugated equine estrogen (CEE), CEE plus medroxyprogesterone acetate (MPA), CEE plus Nomegestrol acetate (NA), and raloxifene on serum high sensitivity C-reactive protein (hs-CRP) and homocysteine (Hcy) levels in healthy postmenopausal women.

Materials: One hundred seven healthy postmenopausal women were recruited in a prospective, randomized, and placebo-controlled 6 months study. Of these, 18 were hysterectomized and received daily oral 0.625 mg CEE. Eighty nine non-hysterectomized women were randomly allocated to one of four groups: a group (22 patients) treated with CEE, 0.625 mg/daily plus MPA 2.5 mg/daily; a group (22 patients) treated with CEE, 0.625 mg/daily plus NA 5 mg/daily; a group (23 patients) treated with raloxifene hydrochloride, 60 mg once daily; and a placebo group (22 patients). Hcy and hs-CRP were measured at baseline and at 3 and 6 months.

Results: CEE (20%, P=0.03) and CEE+MPA (59%, P=0.006) increased serum hs-CRP levels significantly, whereas CEE+NA decreased serum hs-CRP by 25% (P=0.01). Raloxifene had no significant effect on serum hs-CRP levels during and after the treatment. In all active treatment groups serum Hcy levels decreased significantly compared to baseline and placebo.

Conclusions: Conjugated equine estrogen, hormone replacement therapies, and raloxifene lower serum Hcy levels to a comparable extent in postmenopausal women. Hs-CRP, as a cardiovascular risk factor, is not influenced by raloxifene, whereas CEE and CEE plus MPA significantly increase hs-CRP levels. Treatment with CEE plus NA reduces serum hs-CRP levels.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • C-Reactive Protein / analysis
  • C-Reactive Protein / drug effects*
  • Drug Combinations
  • Estrogen Replacement Therapy*
  • Estrogens, Conjugated (USP) / administration & dosage
  • Estrogens, Conjugated (USP) / pharmacology*
  • Female
  • Homocysteine / blood
  • Homocysteine / drug effects*
  • Humans
  • Medroxyprogesterone Acetate / administration & dosage
  • Medroxyprogesterone Acetate / pharmacology
  • Megestrol / administration & dosage
  • Megestrol / pharmacology
  • Middle Aged
  • Norpregnadienes / administration & dosage
  • Norpregnadienes / pharmacology
  • Postmenopause / blood
  • Prospective Studies
  • Raloxifene Hydrochloride / administration & dosage
  • Raloxifene Hydrochloride / pharmacology*
  • Selective Estrogen Receptor Modulators / administration & dosage
  • Selective Estrogen Receptor Modulators / pharmacology*
  • Treatment Outcome

Substances

  • Drug Combinations
  • Estrogens, Conjugated (USP)
  • Norpregnadienes
  • Selective Estrogen Receptor Modulators
  • Homocysteine
  • Raloxifene Hydrochloride
  • nomegestrol acetate
  • C-Reactive Protein
  • Medroxyprogesterone Acetate
  • Megestrol