Depression of hepatic drug metabolism in endotoxin-treated and sarcoma-bearing mice

Res Commun Chem Pathol Pharmacol. 1992 May;76(2):223-31.

Abstract

The effect of a single dose of bacterial endotoxin (lipopolysaccharide, LPS) was compared with that of tumor implantation in mice on the activity of several hepatic cytochrome P-450-dependent monooxygenases. These included ethoxycoumarin O-deethylase, p-nitrophenol hydroxylase, aminopyrine N-demethylase, pentoxyresorufin O-depentylase, ethoxyresorufin O-deethylase and testosterone hydroxylase. For this purpose, mice were treated i.p. with 5 micrograms of LPS or implanted in the right paw with S 180 sarcoma. A comparable depression (30-50%) of total microsomal P-450 content as well as of the different P-450 monooxygenase activities tested was observed in LPS-treated mice (24 h after LPS) and in tumor bearing mice (12 days after implantation). The lack of differences in the pattern of depression of microsomal enzymes between LPS-treated and tumor-bearing mice suggests that a common mechanisms might be involved in the depression of P-450 by LPS or S-180 implantation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Body Weight / drug effects
  • Cytochrome P-450 Enzyme System / metabolism
  • Depression, Chemical
  • Eating / drug effects
  • Escherichia coli / metabolism*
  • Lipopolysaccharides*
  • Liver / drug effects
  • Liver / enzymology
  • Liver / metabolism*
  • Male
  • Mice
  • Microsomes, Liver / drug effects
  • Microsomes, Liver / enzymology
  • Mixed Function Oxygenases / metabolism
  • Pharmaceutical Preparations / metabolism*
  • Sarcoma 180 / metabolism*
  • Testosterone / metabolism

Substances

  • Lipopolysaccharides
  • Pharmaceutical Preparations
  • Testosterone
  • Cytochrome P-450 Enzyme System
  • Mixed Function Oxygenases