Regulation of blood glucose by hypothalamic pyruvate metabolism

Science. 2005 Aug 5;309(5736):943-7. doi: 10.1126/science.1112085.

Abstract

The brain keenly depends on glucose for energy, and mammalians have redundant systems to control glucose production. An increase in circulating glucose inhibits glucose production in the liver, but this negative feedback is impaired in type 2 diabetes. Here we report that a primary increase in hypothalamic glucose levels lowers blood glucose through inhibition of glucose production in rats. The effect of glucose requires its conversion to lactate followed by stimulation of pyruvate metabolism, which leads to activation of adenosine triphosphate (ATP)-sensitive potassium channels. Thus, interventions designed to enhance the hypothalamic sensing of glucose may improve glucose homeostasis in diabetes.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Astrocytes / metabolism
  • Blood Glucose / metabolism*
  • Citric Acid Cycle
  • Feedback, Physiological
  • Glucose / administration & dosage
  • Glucose / metabolism*
  • Glucose-6-Phosphatase / metabolism
  • Hypothalamus / metabolism*
  • Injections, Intraventricular
  • Lactic Acid / metabolism
  • Liver / metabolism*
  • Male
  • Neurons / metabolism
  • Potassium Channels / metabolism
  • Pyruvates / metabolism*
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Blood Glucose
  • Potassium Channels
  • Pyruvates
  • Lactic Acid
  • Glucose-6-Phosphatase
  • Glucose