Semisynthetic tellurosubtilisin with glutathione peroxidase activity

J Am Chem Soc. 2005 Aug 24;127(33):11588-9. doi: 10.1021/ja052451v.

Abstract

Reaction of the hydroxyl group of serine-221 of subtilisin with phenylmethanesulfonylfluoride followed by nucleophilic substitution with sodium hydrogen telluride, a semisynthetic telluroprotein, tellurosubtilisin, was prepared. Tellurosubtilisin, which displays high substrate specificity for aromatic thiols, exhibits remarkable peroxidase activity and catalyzes the reduction of hydrogen peroxide by 3-carboxy-4-nitrobenzenethiol 20 000 times more efficiently than diphenyl diselenide.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Catalysis
  • Glutathione Peroxidase / chemistry*
  • Subtilisin / chemical synthesis*
  • Subtilisin / chemistry
  • Tellurium / chemistry

Substances

  • Glutathione Peroxidase
  • Subtilisin
  • Tellurium