BEL-1, a novel clavulanic acid-inhibited extended-spectrum beta-lactamase, and the class 1 integron In120 in Pseudomonas aeruginosa

Antimicrob Agents Chemother. 2005 Sep;49(9):3743-8. doi: 10.1128/AAC.49.9.3743-3748.2005.

Abstract

Screening by a double-disk synergy test identified a Pseudomonas aeruginosa isolate that produced a clavulanic acid-inhibited expanded-spectrum beta-lactamase (ESBL). Cloning and sequencing identified a novel ESBL, BEL-1, weakly related to other Ambler class A ESBLs. beta-Lactamase BEL-1 hydrolyzed significantly most expanded-spectrum cephalosporins and aztreonam, and its activity was inhibited by clavulanic acid, tazobactam, cefoxitin, moxalactam, and imipenem. This chromosome-encoded ESBL gene was embedded in a class 1 integron containing three other gene cassettes. In addition, this integron was bracketed by Tn1404 transposon sequences at its right end and by P. aeruginosa-specific sequences at its left end.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Anti-Bacterial Agents / pharmacology*
  • Clavulanic Acid / pharmacology*
  • Cloning, Molecular
  • DNA, Bacterial / genetics
  • Enzyme Inhibitors / pharmacology*
  • Genes, Bacterial / genetics*
  • Integrons / genetics*
  • Isoelectric Focusing
  • Kinetics
  • Microbial Sensitivity Tests
  • Molecular Sequence Data
  • Plasmids / genetics
  • Pseudomonas aeruginosa / drug effects*
  • Pseudomonas aeruginosa / genetics*
  • Reverse Transcriptase Polymerase Chain Reaction
  • Spectrophotometry, Ultraviolet
  • beta-Lactamase Inhibitors
  • beta-Lactamases / genetics*
  • beta-Lactamases / metabolism

Substances

  • Anti-Bacterial Agents
  • DNA, Bacterial
  • Enzyme Inhibitors
  • beta-Lactamase Inhibitors
  • Clavulanic Acid
  • beta-Lactamases
  • beta-lactamase BEL-1, Pseudomonas aeruginosa