Beclomethasone dipropionate attenuates airways hyperresponsiveness to neurokinin A and histamine in asthma

Respir Med. 2006 Jun;100(6):1006-12. doi: 10.1016/j.rmed.2005.09.038. Epub 2005 Nov 15.

Abstract

Background: Inhaled corticosteroids (ICS) are the most effective anti-inflammatory agents available for the treatment of asthma but they produce only modest effects on airway inflammation and non-specific bronchial hyperresponsiveness (BHR). However, little is known about the possibility that treatment with ICS might cause additional protection on BHR to inhaled tachykinins such as neurokinin A (NKA).

Objective: Therefore, we compared the effects of beclomethasone dipropionate (BDP) on the degree of BHR to inhaled histamine and NKA in a double-blind, controlled, cross-over study of asthmatic patients.

Methods: Patients attended the laboratory before and after each 6 weeks treatment period to undertake concentration-response studies with histamine and NKA. Bronchial responsiveness to both funs was expressed as the provocative concentration producing a 20% decrease in FEV(1) from baseline (PC(20)).

Results: BDP therapy attenuated the constrictor response to both agonists to a similar degree, their geometric mean (range) PC(20) values increasing from 0.47 (0.21-1.41) mg/ml to 2.43 (0.51-4.50) mg/ml (P<0.01, post-salb vs. post-BDP treatment) and from 101.7 (27.3-356.1) microg/ml to 666.7 (151.5-1,000) microg/ml (P<0.01, post-salb vs. post-BDP treatment) for histamine and NKA, respectively.

Conclusion: Airway responsiveness to histamine and NKA is reduced by BDP to the same extent. As a result of these findings, provocation with NKA is unlikely to provide additional useful information in the assessment of airway inflammation in asthma.

Publication types

  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Inhalation
  • Adrenal Cortex Hormones / pharmacology*
  • Adrenal Cortex Hormones / therapeutic use
  • Adrenergic beta-Agonists / therapeutic use
  • Adult
  • Albuterol / therapeutic use
  • Analysis of Variance
  • Asthma / drug therapy
  • Asthma / physiopathology*
  • Beclomethasone / pharmacology*
  • Beclomethasone / therapeutic use
  • Bronchial Hyperreactivity / physiopathology
  • Bronchial Provocation Tests
  • Cross-Over Studies
  • Dose-Response Relationship, Drug
  • Double-Blind Method
  • Female
  • Histamine
  • Humans
  • Male
  • Neurokinin A
  • Statistics, Nonparametric

Substances

  • Adrenal Cortex Hormones
  • Adrenergic beta-Agonists
  • Histamine
  • Neurokinin A
  • Beclomethasone
  • Albuterol