Tumor angiogenic vasculature targeting with PAMAM dendrimer-RGD conjugates

Chem Commun (Camb). 2005 Dec 14:(46):5739-41. doi: 10.1039/b507350b. Epub 2005 Oct 10.

Abstract

PAMAM dendrimer-RGD-4C peptide conjugate was synthesized and in vitro targeting efficacy to integrin receptor expressing cells was studied by flow cytometry and confocal microscopy.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Angiogenesis Inhibitors / chemistry*
  • Angiogenesis Inhibitors / metabolism*
  • Animals
  • Cell Line
  • Dendrimers
  • Drug Delivery Systems / methods*
  • Humans
  • Integrins / metabolism
  • Mice
  • Molecular Structure
  • Neoplasms / blood supply*
  • Neoplasms / drug therapy*
  • Neovascularization, Pathologic
  • Oligopeptides / chemistry
  • Oligopeptides / metabolism*
  • Polyamines / chemistry
  • Polyamines / metabolism*

Substances

  • Angiogenesis Inhibitors
  • Dendrimers
  • Integrins
  • Oligopeptides
  • PAMAM Starburst
  • Polyamines
  • arginyl-glycyl-aspartic acid