Influence of the hemoglobin solution HBOC-201 on tissue oxygenation in the rat R1H-tumor

Artif Cells Blood Substit Immobil Biotechnol. 2005;33(4):379-89. doi: 10.1080/10731190500289750.

Abstract

Background: HBOC-201 is an ultra purified bovine hemoglobin solution. It has already been used in clinical phase II/III trials for emergency treatments. Animal experiments have shown that HBOC-201 is highly effective in tissue oxygenation. The study was performed in order to assess the potential of low dose HBOC-201 to improve tumor oxygenation.

Methods: 30 rats with a subcutaneously growing rhabdomyosarcoma R1H tumor were randomly assigned either to be ventilated with carbogen (n = 10), or to receive an IV injection of 0.3 g/kg HBOC-201 (n = 10) or a combination of 0.3 g/kg HBOC-201 and carbogen breathing (n = 10). Under general anesthesia the effects of the respective treatment on the tissue oxygen tension (tpO2) of the tumor were determined using a flexible stationary probe at baseline (b) and 15 and 60 min after application of the respective medication.

Results: HBOC-201 alone failed to improve tumor tpO2 (b: 1.3 +/- 1.2mmHg; 15min: 1.4 +/- 1 mmHg; 60min: 1 +/- 1 mmHg). In combination with carbogen the mean tpO2 of the tumor raised in comparison to baseline values (b: 3.1 +/- 4.6 mmHg; mmHg; 15min: 8.5 +/- 11*mmHg; 60min: 4.8 +/- 5mmHg; *p < 0.05 vs. b), but this effect was less pronounced than the increase in tpO2 by carbogen alone (b: 3.4 +/- 3.4mmHg; 15min: 9 +/- 10* mmHg; 60 min: 13 +/- 19* mmHg; *p < 0.05 vs. b).

Conclusion: The application of low dose hemoglobin solution HBOC-201 does not result in improvement of tissue oxygenation in the rat rhabdomyosarcoma R1H.

MeSH terms

  • Animals
  • Blood Substitutes / administration & dosage
  • Blood Substitutes / pharmacology
  • Carbon Dioxide / administration & dosage
  • Carbon Dioxide / pharmacology
  • Drug Evaluation, Preclinical
  • Hemoglobins / administration & dosage
  • Hemoglobins / pharmacology*
  • Hypoxia / drug therapy
  • Oxygen / administration & dosage
  • Oxygen / metabolism*
  • Oxygen / pharmacology
  • Rats
  • Rhabdomyosarcoma / metabolism*
  • Rhabdomyosarcoma / pathology
  • Tissue Distribution / drug effects

Substances

  • Blood Substitutes
  • Hemoglobins
  • Carbon Dioxide
  • HBOC 201
  • carbogen
  • Oxygen