Prostaglandin (PG) E1 and 13,14-dihydro (DH) PGE1 are diminishing radiation-induced arterial damage

Agents Actions Suppl. 1992:37:58-65. doi: 10.1007/978-3-0348-7262-1_9.

Abstract

Rabbit abdominal aorta was irradiated with single or repeated doses up to 10 Gy. The rabbits were killed at different time intervals after irradiation. 5 micrograms/kg x 6/hr PGE1 or its biologically active metabolite 13,14-DH-PGE1 were administered either 6 hours before or 6 hours after irradiation. The administration of both PGEs reduced radiation-induced mitotic activity (3H-thymidine incorporation) and extracellular matrix [collagen-(14C-proline) and glycosaminoglycan (35-S-sulphate)]-formation as determined by means of autoradiography. The initial peak increase in vascular PGI2-synthesis was partly abolished, while the long lasting depression was less pronounced. 13,14-DH-PGE1 was only slightly less active as compared to the parent compound. Pre-radiation treatment was more effective than post-irradiation therapy. These findings suggest that both the PGs exert significant radiation-protective actions on the arterial wall.

MeSH terms

  • Alprostadil / analogs & derivatives*
  • Alprostadil / pharmacology*
  • Animals
  • Aorta, Abdominal / drug effects
  • Aorta, Abdominal / radiation effects
  • Arteries / radiation effects*
  • Autoradiography
  • Dose-Response Relationship, Radiation
  • Extracellular Matrix / drug effects
  • Extracellular Matrix / radiation effects
  • Male
  • Mitosis / drug effects
  • Mitosis / radiation effects
  • Rabbits
  • Radiation Injuries, Experimental / prevention & control*
  • Radiation-Protective Agents / pharmacology*

Substances

  • Radiation-Protective Agents
  • 13,14-dihydroprostaglandin E1
  • Alprostadil