Dichotomous but stringent substrate selection by the dual-function Cdk7 complex revealed by chemical genetics

Nat Struct Mol Biol. 2006 Jan;13(1):55-62. doi: 10.1038/nsmb1028. Epub 2005 Dec 4.

Abstract

Cdk7 performs two essential but distinct functions as a CDK-activating kinase (CAK) required for cell-cycle progression and as the RNA polymerase II (Pol II) CTD kinase of general transcription factor IIH. To investigate the substrate specificity underlying this dual function, we created an analog-sensitive (AS) Cdk7 able to use bulky ATP derivatives. Cdk7-AS-cyclin H-Mat1 phosphorylates approximately 10-15 endogenous polypeptides in nuclear extracts. We identify seven of these as known and previously unknown Cdk7 substrates that define two classes: proteins such as Pol II and transcription elongation factor Spt5, recognized efficiently only by the fully activated Cdk7 complex, through sequences surrounding the site of phosphorylation; and CDKs, targeted equivalently by all active forms of Cdk7, dependent on substrate motifs remote from the phosphoacceptor residue. Thus, Cdk7 accomplishes dual functions in cell-cycle control and transcription not through promiscuity but through distinct, stringent modes of substrate recognition.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / analogs & derivatives
  • Adenosine Triphosphate / pharmacology
  • Amino Acid Sequence
  • Cell Extracts
  • Cell Nucleus / metabolism
  • Conserved Sequence
  • Cyclin-Dependent Kinase-Activating Kinase
  • Cyclin-Dependent Kinases / chemistry*
  • Cyclin-Dependent Kinases / genetics
  • Cyclin-Dependent Kinases / metabolism*
  • Enzyme Activation
  • HeLa Cells
  • Humans
  • Molecular Sequence Data
  • Phosphorylation
  • Protein Binding
  • Sequence Alignment
  • Substrate Specificity

Substances

  • Cell Extracts
  • Adenosine Triphosphate
  • Cyclin-Dependent Kinases
  • Cyclin-Dependent Kinase-Activating Kinase
  • CDK7 protein, human