Ion-binding properties of the ClC chloride selectivity filter

EMBO J. 2006 Jan 11;25(1):24-33. doi: 10.1038/sj.emboj.7600909. Epub 2005 Dec 8.

Abstract

The ClC channels are members of a large protein family of chloride (Cl-) channels and secondary active Cl- transporters. Despite their diverse functions, the transmembrane architecture within the family is conserved. Here we present a crystallographic study on the ion-binding properties of the ClC selectivity filter in the close homolog from Escherichia coli (EcClC). The ClC selectivity filter contains three ion-binding sites that bridge the extra- and intracellular solutions. The sites bind Cl- ions with mM affinity. Despite their close proximity within the filter, the three sites can be occupied simultaneously. The ion-binding properties are found conserved from the bacterial transporter EcClC to the human Cl- channel ClC-1, suggesting a close functional link between ion permeation in the channels and active transport in the transporters. In resemblance to K+ channels, ions permeate the ClC channel in a single file, with mutual repulsion between the ions fostering rapid conduction.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bromine / chemistry
  • Cations, Monovalent / chemistry
  • Chloride Channels / chemistry*
  • Chloride Channels / genetics
  • Chlorine / chemistry
  • Crystallography, X-Ray
  • Escherichia coli Proteins / chemistry*
  • Escherichia coli Proteins / genetics
  • Humans
  • Mutation
  • Protein Conformation

Substances

  • Cations, Monovalent
  • Chloride Channels
  • ClC protein, E coli
  • Escherichia coli Proteins
  • Chlorine
  • Bromine

Associated data

  • PDB/2EXW
  • PDB/2EXY
  • PDB/2EZ0