Abstract
It has been reported that collagen II (CII)-derived peptide induced T-cell activation via its amino acids responsible for T-cell receptor (TCR) recognition. In this study, three altered CII263-272 peptide ligands (APL) containing multiple substitutions of TCR contact residues were synthesized. Their roles in inhibition of T-cell activation were evaluated in peripheral blood lymphocytes (PBL) of rheumatoid arthritis (RA) in vitro. It was shown that 41% (25/61) of RA patients were responsive to the wild-type antigenic CII263-272. In contrast, marginal or silent T-cell responses to the three APLs were found, accompanied by inhibitory effects on secretion of Th1 type cytokines and expression of cell surface markers, CD69 and CD25. In addition, T-cell activation induced by the wild-type antigenic CII263-272 was inhibited by all the three APLs in a dose-dependent manner. It is demonstrated that APLs with substitutions of TCR contact residues are capable of down-regulating T-cell responses in PBLs of RA, suggesting that the CII-derived APLs are potentially therapeutic in RA.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Adult
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Aged
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Antigens, CD / biosynthesis
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Antigens, CD / genetics
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Antigens, Differentiation, T-Lymphocyte / biosynthesis
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Antigens, Differentiation, T-Lymphocyte / genetics
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Arthritis, Rheumatoid / immunology*
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CD4-Positive T-Lymphocytes / metabolism
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Cell Proliferation
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Cells, Cultured
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Collagen Type II / immunology*
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Collagen Type II / metabolism
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Cytokines / metabolism
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Female
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HLA-DR4 Antigen / immunology
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HLA-DR4 Antigen / metabolism
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Humans
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Immunosuppressive Agents / pharmacology*
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Lectins, C-Type
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Ligands
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Lymphocyte Activation / immunology*
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Male
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Middle Aged
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Peptide Fragments / immunology*
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Peptide Fragments / metabolism
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Receptors, Antigen, T-Cell / immunology
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Receptors, Antigen, T-Cell / metabolism
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Receptors, Interleukin-2 / biosynthesis
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Receptors, Interleukin-2 / genetics
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T-Lymphocytes / immunology*
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T-Lymphocytes / metabolism
Substances
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Antigens, CD
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Antigens, Differentiation, T-Lymphocyte
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CD69 antigen
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Collagen Type II
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Cytokines
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HLA-DR4 Antigen
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Immunosuppressive Agents
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Lectins, C-Type
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Ligands
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Peptide Fragments
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Receptors, Antigen, T-Cell
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Receptors, Interleukin-2