Asparagine depletion after pegylated E. coli asparaginase treatment and induction outcome in children with acute lymphoblastic leukemia in first bone marrow relapse: a Children's Oncology Group study (CCG-1941)

Pediatr Blood Cancer. 2006 Aug;47(2):141-6. doi: 10.1002/pbc.20713.

Abstract

Purpose: Re-induction outcomes vary for children with acute lymphoblastic leukemia (ALL) and marrow relapse. We explored possible relationships among asparaginase (ASNase) activity levels, asparagine (ASN) depletion, anti-ASNase antibody titers, and response to re-induction therapy in children and adolescents with ALL and an 'early' first marrow relapse.

Patients and methods: After appropriate informed consent, we enrolled children and adolescents 1-21 years old with ALL and first marrow relapse within 12 months of completion of primary therapy. Induction therapy included intramuscular pegylated ASNase on Days 2 and 16. We assessed ASNase activity, anti-ASNase antibody titers against native and pegylated (E. coli) ASNase, and amino acid levels of asparagine (ASN) and glutamine (GLN) on Days 0, 14, and 35 of re-induction.

Results: Ninety-three patients were at least partially assessable. Among 21 patients with M1 marrow status at Day 35, the median Day 14 ASN level was <1 microM. This is significantly lower than the median Day 14 ASN level of 4 microM in the group of patients with M3 marrow at Day 35. Neither Day 0 nor Day 35 antibody titers predicted ASNase enzymatic activity level on Day 14. Surprisingly, Day 14 ASNase activity did not predict serum ASN level on Day 14. However, Day 0 and Day 35 anti-native ASNase antibody titers, and Day 0 anti-PEG ASNase antibody titers correlated positively with Day 14 serum ASN levels as one might expect from neutralizing antibody. Day 35 anti-PEG ASNase antibody titers did not.

Conclusions: Patients with greater ASN depletion were more likely to achieve second remission in the context of six-drug therapy.

Publication types

  • Clinical Conference

MeSH terms

  • Antibody Formation / drug effects
  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents / pharmacology*
  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use
  • Asparaginase / administration & dosage
  • Asparaginase / immunology
  • Asparaginase / pharmacology*
  • Asparagine / drug effects*
  • Asparagine / metabolism
  • Child
  • Female
  • Glutamic Acid / drug effects
  • Glutamic Acid / metabolism
  • Humans
  • Injections, Intramuscular
  • Male
  • Polyethylene Glycols / administration & dosage
  • Polyethylene Glycols / pharmacology*
  • Precursor Cell Lymphoblastic Leukemia-Lymphoma / drug therapy*
  • Precursor Cell Lymphoblastic Leukemia-Lymphoma / pathology
  • Recurrence
  • Remission Induction
  • Statistics, Nonparametric

Substances

  • Antineoplastic Agents
  • Glutamic Acid
  • Polyethylene Glycols
  • Asparagine
  • pegaspargase
  • Asparaginase