Imatinib mesylate minimally affects bcr-abl+ and normal monocyte-derived dendritic cells but strongly inhibits T cell expansion despite reciprocal dendritic cell-T cell activation

J Leukoc Biol. 2006 Apr;79(4):747-56. doi: 10.1189/jlb.0705419. Epub 2006 Feb 3.

Abstract

In chronic myeloid leukemia, bcr-abl+ monocytes provide a unique opportunity to generate dendritic cells (DC) expressing a broad spectrum of leukemic antigens, and bcr-abl+ DC vaccines may allow immunological eradication of leukemic cells persisting under treatment with the tyrosine kinase inhibitor imatinib. However, the efficiency of bcr-abl+ DC vaccines will critically depend on the absence of deleterious effects of bcr-abl and of imatinib on DC functions. We show that bcr-abl+ monocytes, devoid of contamination of CD14low granulocytic precursors, differentiate into DC with typical immunophenotypical and functional features, and bcr-abl transcription decreases simultaneously. During differentiation, imatinib induces a slight increase of DC apoptosis and prevents CD1a up-regulation in a dose-dependent manner in bcr-abl+ and normal monocyte-derived DC, but at most, 25% of DC fail to acquire CD1a. When DC maturation is induced in the presence of imatinib, bcr-abl+ and normal monocyte-derived DC up-regulate major histocompatibility complex and costimulatory molecules, CC chemokine receptor 7 and CD83. However, secretion of interleukin-12p70 is decreased in a dose-dependent manner. Imatinib exposure of bcr-abl+ and normal monocyte-derived DC during differentiation and maturation is not detrimental to T cell immunostimulatory functions of DC. In sharp contrast, imatinib, when added to DC-T cell cultures, profoundly suppresses DC-mediated T cell proliferation, despite reciprocal DC-T cell activation attested by up-regulation of CD25 on T cells and of CD86 on DC. Our findings demonstrate that T cells, not normal or bcr-abl+ monocyte-derived DC, are major targets for imatinib immunomodulatory effects. It can be envisioned already that imatinib-free windows will be required to enable vaccination-induced, leukemia-specific T cell expansion.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Benzamides
  • Cell Differentiation / immunology
  • Cell Division / drug effects
  • Cell Division / immunology
  • Coculture Techniques
  • Dendritic Cells / drug effects*
  • Dendritic Cells / immunology
  • Fusion Proteins, bcr-abl / drug effects*
  • Fusion Proteins, bcr-abl / immunology
  • Humans
  • Imatinib Mesylate
  • Immunologic Tests
  • Interleukin-12 / metabolism
  • Lymphocyte Activation / drug effects
  • Lymphocyte Activation / immunology*
  • Monocytes / drug effects*
  • Monocytes / immunology
  • Phenotype
  • Piperazines / pharmacology*
  • Pyrimidines / pharmacology*
  • T-Lymphocytes / drug effects*
  • T-Lymphocytes / immunology
  • Time Factors

Substances

  • Benzamides
  • Piperazines
  • Pyrimidines
  • Interleukin-12
  • Imatinib Mesylate
  • Fusion Proteins, bcr-abl