The two isotypes of the human insulin receptor (HIR-A and HIR-B) follow different internalization kinetics

Biochem Biophys Res Commun. 1991 Jun 28;177(3):1013-8. doi: 10.1016/0006-291x(91)90639-o.

Abstract

Human insulin receptor (HIR) is expressed in two isoforms which differ in the C-terminal end of the alpha-subunit (HIR-A = -12 aa, HIR-B = +12 aa). We studied internalization kinetics of HIR-A and HIR-B in Rat1 fibroblasts. Internalized receptors were quantified by 125I-insulin binding after cell trypsinisation and solubilization, surface receptors were determined by 125I-insulin binding to intact cells and by chemical crosslinking with B26-125I-insulin. HIR-A and HIR-B show different kinetics of receptor internalization. While in HIR-A cells the maximum of internalization (approx. 65% of total) is reached after 10 min followed by a high recycling rate (approx. 80% of internalized receptors after 20 min), the internalization in HIR-B cells reaches a maximum (approx. 60% of total) after 15 min without detectable recycling within 30 min. The data show that the different alpha-subunits of both receptor types determine different velocities of internalization and determine whether a fast recycling occurs.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Cell Line
  • Cell Membrane / metabolism
  • Humans
  • Insulin / metabolism
  • Isoenzymes / metabolism
  • Kinetics
  • Macromolecular Substances
  • Phosphorylation
  • Protein-Tyrosine Kinases / metabolism
  • Rats
  • Receptor, Insulin / genetics
  • Receptor, Insulin / metabolism*
  • Transfection

Substances

  • Insulin
  • Isoenzymes
  • Macromolecular Substances
  • Protein-Tyrosine Kinases
  • Receptor, Insulin