Tris(pyrone) chelates of Gd(III) as high solubility MRI-CA

J Am Chem Soc. 2006 Feb 22;128(7):2222-3. doi: 10.1021/ja057954f.

Abstract

Two tripodal, hexadentate pyrone-based chelators have been prepared. These ligands form stable, soluble complexes with gadolinium(III). The complexes show aqueous stability comparable to that of [Gd(DTPA)]2- at pH 7.4. Evaluation by relaxometry shows that these complexes have two inner-sphere water molecules and a very fast water exchange rate. The solution behavior of these complexes suggests that they may be attractive as high relaxivity, next-generation magnetic resonance imaging contrast agents.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Chelating Agents / chemical synthesis
  • Chelating Agents / chemistry*
  • Contrast Media / chemical synthesis
  • Contrast Media / chemistry*
  • Ethylenediamines / chemistry
  • Gadolinium / chemistry*
  • Magnetic Resonance Imaging / methods*
  • Pyrones / chemical synthesis
  • Pyrones / chemistry*
  • Solubility

Substances

  • Chelating Agents
  • Contrast Media
  • Ethylenediamines
  • Pyrones
  • tris(2-aminoethyl)amine
  • Gadolinium