Effect of co-dergocrine in the autoperfused superior mesenteric vascular bed of the rat

J Auton Pharmacol. 1991 Jun;11(3):155-65. doi: 10.1111/j.1474-8673.1991.tb00315.x.

Abstract

1. The influence of local administration of co-dergocrine in the in situ, constant flow autoperfused, superior mesenteric vascular bed of the rat was investigated. 2. Local infusion of co-dergocrine (0.1 micrograms kg-1 min-1) reduced the pressor response to electrical stimulation of the periarterial sympathetic nerves for the whole frequency range studied during cumulative frequency-response curves (1-8 Hz). 3. Co-dergocrine (0.01, 0.03, 0.1 micrograms kg-1 min-1) dose-dependently inhibited the pressor response to electrical stimulation at 4 Hz; increases in perfusion pressure produced by locally administered noradrenaline were inhibited to the same degree. 4. Pressor responses induced by locally administered phenylephrine were also inhibited by co-dergocrine (0.1 micrograms kg-1 min-1) while those produced by local injection of angiotensin II were not. 5. Local administration of the DA1-/DA2-receptor antagonist haloperidol (1 microgram kg-1), the DA2-receptor antagonist domperidone (10 micrograms kg-1) and the alpha 2-adrenoceptor antagonist rauwolscine (100 micrograms kg-1) partially prevented the influence of co-dergocrine on the electrically induced response. 6. The results show that the effect of co-dergocrine in the rat superior mesenteric vascular bed cannot simply be ascribed to interaction with the presynaptic inhibitory DA2-receptors on the noradrenergic nerve endings; it also has an antagonistic action at the postsynaptic alpha 1-adrenoceptors and an agonist action at the presynaptic alpha 2-adrenoceptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiotensin II / antagonists & inhibitors
  • Animals
  • Dihydroergotoxine / administration & dosage
  • Dihydroergotoxine / antagonists & inhibitors
  • Dihydroergotoxine / pharmacology*
  • Domperidone / pharmacology
  • Female
  • Haloperidol / pharmacology
  • Male
  • Mesenteric Veins / drug effects*
  • Norepinephrine / antagonists & inhibitors
  • Perfusion / methods
  • Phenylephrine / antagonists & inhibitors
  • Rats
  • Rats, Inbred Strains
  • Receptors, Adrenergic, alpha / metabolism
  • Yohimbine / pharmacology

Substances

  • Receptors, Adrenergic, alpha
  • Dihydroergotoxine
  • Angiotensin II
  • Phenylephrine
  • Yohimbine
  • Domperidone
  • Haloperidol
  • Norepinephrine