The inhibitory effects of oxytocin on distal colonic contractile activity in rabbits are enhanced by ovarian steroids

Acta Physiol (Oxf). 2006 Feb;186(2):141-9. doi: 10.1111/j.1365-201X.2005.01506.x.

Abstract

Aims: To study the effects of oxytocin on isolated rabbit distal colon and the regulation of ovarian steroids by its action.

Methods: Muscle strips parallel to either the circular or the longitudinal fibres were excised and suspended in tissue chambers containing 5 mL Krebs solution (37 degrees C) and bubbled continuously with 95% O(2) and 5% CO(2). The effects of oxytocin on isometric spontaneous contractile responses were recorded. The effects of atosiban, tetrodotoxin, Mg(2+), progesterone and oestradiol on the oxytocin-induced response were also examined.

Results: Oxytocin (1, 10 and 100 nmol L(-1)) dose dependently decreased the area under the contraction curve of distal colonic smooth muscle strips. The oxytocin receptor antagonist atosiban blocked the oxytocin (10 nmol L(-1))-caused responses in a dose-dependent manner. Tetrodotoxin (10 micromol L(-1)) had no effect on the oxytocin-induced response. Mg(2+)-free Krebs solution attenuated the oxytocin-induced response, but oestradiol (0.1 micromol L(-1)) or progesterone (0.1 micromol L(-1)) increased the oxytocin-induced response.

Conclusion: These results suggest that oxytocin inhibits the contractile motility of the distal colon, which is regulated by Mg(2+) and ovarian steroids.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Colon / drug effects*
  • Colon / physiology
  • Diffusion Chambers, Culture
  • Dose-Response Relationship, Drug
  • Drug Synergism
  • Estradiol / pharmacology
  • Female
  • Gastrointestinal Motility / drug effects
  • Hormone Antagonists / pharmacology
  • Magnesium / pharmacology
  • Muscle Contraction / drug effects*
  • Muscle, Smooth / drug effects*
  • Muscle, Smooth / physiology
  • Oxytocin / antagonists & inhibitors
  • Oxytocin / pharmacology*
  • Progesterone / pharmacology
  • Rabbits
  • Receptors, Oxytocin / antagonists & inhibitors
  • Tetrodotoxin / pharmacology
  • Vasotocin / analogs & derivatives
  • Vasotocin / pharmacology

Substances

  • Hormone Antagonists
  • Receptors, Oxytocin
  • atosiban
  • Tetrodotoxin
  • Progesterone
  • Estradiol
  • Oxytocin
  • Magnesium
  • Vasotocin