Comparison of pharmacological agents (aspartate vs. aminophosphonobutyric plus kynurenic acids) to block synaptic transmission from retinal photoreceptors in frog

Exp Eye Res. 1991 Jun;52(6):691-8. doi: 10.1016/0014-4835(91)90021-6.

Abstract

The combination of aminophosphonobutyric plus kynurenic acids (APB/Kyn) was compared to aspartate with respect to its ability to block synaptic transmission from photoreceptors. Like aspartate, APB/Kyn blocks photoreceptor synaptic transmission, as monitored by the b- and d-waves of the electroretinogram, by the proximal negative response and M-wave of the proximal retina, and by the light-evoked increase in extracellular K+ concentration in the inner plexiform layer. Unlike aspartate, APB/Kyn has relatively minor effects on retinal resistance, light-evoked changes in K+ and Ca2+ concentrations in the subretinal space, light-evoked changes in subretinal space volume, resting extracellular concentrations of K+ and Ca2+ in the proximal and distal retina, and the c-wave. Effects of APB/Kyn are generally more reversible than effects of Asp. A disadvantage of APB/Kyn is that the a-wave usually becomes smaller and slower. Overall, APB/Kyn disrupts the retina less than aspartate. Therefore, in some situations in which blockade of photoreceptor synaptic transmission is desired, the use of APB/Kyn may be preferable to that of aspartate.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Aminobutyrates / pharmacology*
  • Animals
  • Aspartic Acid / pharmacology*
  • Depression, Chemical
  • Electroretinography / drug effects
  • Kynurenic Acid / pharmacology*
  • Photoreceptor Cells / drug effects*
  • Rana pipiens
  • Retina / drug effects*
  • Synaptic Transmission / drug effects*

Substances

  • Aminobutyrates
  • Aspartic Acid
  • Kynurenic Acid
  • 2-amino-4-phosphonobutyric acid