Endocrine and metabolic effects of rosiglitazone in overweight women with PCOS: a randomized placebo-controlled study

Hum Reprod. 2006 Jun;21(6):1400-7. doi: 10.1093/humrep/dei505. Epub 2006 Feb 24.

Abstract

Background: The objective of the study was to assess the therapeutic effects of rosiglitazone in overweight women with polycystic ovary syndrome (PCOS).

Methods: A double-blind, placebo-controlled study was conducted on 30 (BMI > 25 kg/m2, mean age 29.1 +/- 1.2 years) overweight women with PCOS treated with rosiglitazone or placebo for 4 months. Waist-to-hip ratios (WHRs), serum concentrations of sex hormones and binding proteins, blood glucose, serum insulin and serum C-peptide during a 75-g oral glucose tolerance test (OGTT), first-phase insulin secretion as determined by an intravenous glucose tolerance test (IVGTT), M values (expressing insulin sensitivity using a euglycaemic clamp) and calorimetric data were assessed at 0 and 4 months of treatment.

Results: Rosiglitazone improved menstrual cyclicity, increased serum sex hormone-binding globulin (SHBG) levels and decreased serum levels of androstenedione, 17-hydroxyprogesterone (17-OHP), dehydroepiandrosterone (DHEA) and dehydroepiandrosterone sulphate (DHEA-S). Glucose tolerance [expressed as AUC(glucose) during the OGTT] improved (P = 0.002) and peripheral insulin response (expressed as AUC(insulin)) decreased (P = 0.004) in the rosiglitazone group (ROSI group). M value improved in the ROSI group from 33.4 +/- 3.27 to 40.0 +/- 5.51 micromol/kg min (P = 0.04).

Conclusion: Rosiglitazone, by improving menstrual cyclicity, hyperandrogenism, insulin resistance and hyperinsulinaemia, represents an alternative treatment for overweight anovulatory women with PCOS and no pregnancy desire.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 17-alpha-Hydroxyprogesterone / blood
  • Adolescent
  • Adult
  • Area Under Curve
  • Dehydroepiandrosterone / blood
  • Double-Blind Method
  • Female
  • Glucose Tolerance Test
  • Humans
  • Overweight*
  • Placebos
  • Polycystic Ovary Syndrome / complications*
  • Rosiglitazone
  • Sex Hormone-Binding Globulin / biosynthesis
  • Thiazolidinediones / therapeutic use*

Substances

  • Placebos
  • Sex Hormone-Binding Globulin
  • Thiazolidinediones
  • Rosiglitazone
  • Dehydroepiandrosterone
  • 17-alpha-Hydroxyprogesterone