Role of alpha-adrenoceptors in control of plasma potassium in conscious rabbits

J Auton Pharmacol. 1991 Oct;11(5):305-13. doi: 10.1111/j.1474-8673.1991.tb00254.x.

Abstract

1. In conscious fed rabbits the intravenous infusion of amidephrine (10 micrograms kg-1 min-1), an alpha 1-adrenoceptor agonist, caused a significant increase in plasma potassium levels that was blunted by prazosin (50 micrograms kg-1, s.c.). Idazoxan failed to modify this response. 2. Clonidine (2 micrograms kg-1 min-1, i.v.), an alpha 2-adrenoceptor agonist, also evoked a hyperkalaemic response which was antagonized by idazoxan (1 microgram kg-1, s.c.), yohimbine (0.45 mg kg-1, s.c.) and prazosin (50 micrograms kg-1, s.c.). Apamin (40 micrograms kg-1, i.v. bolus) also suppressed the clonidine-mediated hyperkalaemia. 3. Verapamil (5 micrograms kg-1, s.c.) prevented both alpha 1- and alpha 2-adrenoceptor-mediated increase in plasma potassium levels. 4. It is concluded that in conscious fed rabbits both alpha 1- and alpha 2-adrenoceptor stimulation induce hyperkalaemia by activation of hepatic Ca(2+)-activated K(+)-channels.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apamin / pharmacology
  • Calcium Channels / drug effects
  • Calcium Channels / metabolism
  • Clonidine / administration & dosage
  • Clonidine / pharmacology
  • Dioxanes / pharmacology
  • Ethanolamines / administration & dosage
  • Ethanolamines / pharmacology
  • Hyperkalemia / chemically induced
  • Idazoxan
  • Potassium / blood*
  • Prazosin / pharmacology
  • Rabbits
  • Receptors, Adrenergic, alpha / physiology*
  • Verapamil / administration & dosage
  • Verapamil / pharmacology

Substances

  • Calcium Channels
  • Dioxanes
  • Ethanolamines
  • Receptors, Adrenergic, alpha
  • Apamin
  • amidephrine
  • Verapamil
  • Clonidine
  • Potassium
  • Prazosin
  • Idazoxan