LH-RH receptors in the human pancreas. Basis for antihormonal treatment in ductal carcinoma of the pancreas

Int J Pancreatol. 1991 Oct;10(2):151-9.

Abstract

LH-RH-, estrogen-, and progesterone-receptor binding was measured in the human pancreas of patients with ductal pancreatic cancer (n = 23) and chronic pancreatitis (n = 15), and of organ donors (n = 11). Receptor analysis was determined by incubation of the homogenized tissues with estrogen, progesterone, and the LH-RH analog buserelin labeled with iodine-125. Only one biopsy (9%) from normal pancreas had an LH-RH-receptor concentration greater than 3 fmol/mg membrane protein. LH-RH binding levels greater than 3 fmol/mg were detected in 67% of patients with chronic pancreatitis and in 57% of patients with pancreatic cancer. Progesterone levels greater than 15 fmol/mg membrane protein were found in 36% of normal pancreas, in 27% of chronic pancreatitis, and in 17% of pancreatic cancer cases, respectively. The highest concentration of estrogen receptors (greater than 15 fmol/mg membrane protein) was seen in normal pancreas (73%). The increase in LH-RH-receptor concentration in chronic pancreatitis and pancreatic cancer seems to be unspecific, but might be of benefit for antiproliferative treatment in pancreatic cancer.

Publication types

  • Comparative Study

MeSH terms

  • Adult
  • Aged
  • Chronic Disease
  • Estrogens / metabolism
  • Female
  • Gonadotropin-Releasing Hormone / metabolism
  • Humans
  • Male
  • Middle Aged
  • Pancreas / chemistry*
  • Pancreas / metabolism
  • Pancreatic Neoplasms / chemistry*
  • Pancreatic Neoplasms / metabolism
  • Pancreatitis / metabolism*
  • Progesterone / metabolism
  • Radioligand Assay
  • Receptors, Estrogen / analysis
  • Receptors, LHRH / analysis*
  • Receptors, Progesterone / analysis

Substances

  • Estrogens
  • Receptors, Estrogen
  • Receptors, LHRH
  • Receptors, Progesterone
  • Gonadotropin-Releasing Hormone
  • Progesterone