Cyclophilin A renders human immunodeficiency virus type 1 sensitive to Old World monkey but not human TRIM5 alpha antiviral activity

J Virol. 2006 May;80(10):4683-90. doi: 10.1128/JVI.80.10.4683-4690.2006.

Abstract

TRIM5alpha is an important mediator of antiretroviral innate immunity influencing species-specific retroviral replication. Here we investigate the role of the peptidyl prolyl isomerase enzyme cyclophilin A in TRIM5alpha antiviral activity. Cyclophilin A is recruited into nascent human immunodeficiency virus type 1 (HIV-1) virions as well as incoming HIV-1 capsids, where it isomerizes an exposed proline residue. Here we show that cyclophilin A renders HIV-1 sensitive to restriction by TRIM5alpha in cells from Old World monkeys, African green monkey and rhesus macaque. Inhibition of cyclophilin A activity with cyclosporine A, or reducing cyclophilin A expression with small interfering RNA, rescues TRIM5alpha-restricted HIV-1 infectivity. The effect of cyclosporine A on HIV-1 infectivity is dependent on TRIM5alpha expression, and expression of simian TRIM5alpha in permissive feline cells renders them able to restrict HIV-1 in a cyclosporine A-sensitive way. We use an HIV-1 cyclophilin A binding mutant (CA G89V) to show that cyclophilin A has different roles in restriction by Old World monkey TRIM5alpha and owl monkey TRIM-Cyp. TRIM-Cyp, but not TRIM5alpha, recruits its tripartite motif to HIV-1 capsid via cyclophilin A and, therefore, HIV-1 G89V is insensitive to TRIM-Cyp but sensitive to TRIM5alpha. We propose that cyclophilin A isomerization of a proline residue in the TRIM5alpha sensitivity determinant of the HIV-1 capsid sensitizes it to restriction by Old World monkey TRIM5alpha. In humans, where HIV-1 has adapted to bypass TRIM5alpha activity, the effects of cyclosporine A are independent of TRIM5alpha. We speculate that cyclophilin A alters HIV-1 sensitivity to a TRIM5alpha-independent innate immune pathway in human cells.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-HIV Agents / pharmacology*
  • Antiviral Restriction Factors
  • Carrier Proteins / pharmacology*
  • Cats
  • Cell Line
  • Cercopithecidae
  • Cyclophilin A / pharmacology*
  • Cyclosporine / pharmacology
  • Drug Resistance, Viral* / drug effects
  • HIV Infections / drug therapy
  • HIV-1 / drug effects
  • HIV-1 / metabolism*
  • Humans
  • Leukemia Virus, Murine / metabolism
  • Simian Immunodeficiency Virus / metabolism
  • Tripartite Motif Proteins
  • Ubiquitin-Protein Ligases

Substances

  • Anti-HIV Agents
  • Antiviral Restriction Factors
  • Carrier Proteins
  • Tripartite Motif Proteins
  • Cyclosporine
  • TRIM5 protein, human
  • Ubiquitin-Protein Ligases
  • Cyclophilin A