Dietary plant sterols accumulate in the brain

Biochim Biophys Acta. 2006 Apr;1761(4):445-53. doi: 10.1016/j.bbalip.2006.03.015. Epub 2006 Apr 19.

Abstract

Dietary plant sterols and cholesterol have a comparable chemical structure. It is generally assumed that cholesterol and plant sterols do not cross the blood-brain barrier, but quantitative data are lacking. Here, we report that mice deficient for ATP-binding cassette transporter G5 (Abcg5) or Abcg8, with strongly elevated serum plant sterol levels, display dramatically increased (7- to 16-fold) plant sterol levels in the brain. Apolipoprotein E (ApoE)-deficient mice also displayed elevated serum plant sterol levels, which was however not associated with significant changes in brain plant sterol levels. Abcg5- and Abcg8-deficient mice were found to carry circulating plant sterols predominantly in high-density lipoprotein (HDL)-particles, whereas ApoE-deficient mice accommodated most of their serum plant sterols in very low-density lipoprotein (VLDL)-particles. This suggests an important role for HDL and/or ApoE in the transfer of plant sterols into the brain. Moreover, sitosterol upregulated apoE mRNA and protein levels in astrocytoma, but not in neuroblastoma cells, to a higher extend than cholesterol. In conclusion, dietary plant sterols pass the blood-brain barrier and accumulate in the brain, where they may exert brain cell type-specific effects.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily G, Member 5
  • ATP Binding Cassette Transporter, Subfamily G, Member 8
  • ATP-Binding Cassette Transporters / genetics
  • ATP-Binding Cassette Transporters / metabolism
  • Animals
  • Apolipoproteins E / genetics
  • Apolipoproteins E / metabolism
  • Blood-Brain Barrier / physiology
  • Brain / metabolism*
  • Brain Chemistry
  • Cell Line
  • Cholesterol / chemistry
  • Cholesterol / metabolism*
  • Cholesterol, Dietary*
  • Lipoproteins / genetics
  • Lipoproteins / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Phytosterols / chemistry
  • Phytosterols / metabolism*
  • Plants / chemistry*
  • RNA, Messenger / metabolism

Substances

  • ABCG5 protein, mouse
  • ABCG8 protein, mouse
  • ATP Binding Cassette Transporter, Subfamily G, Member 5
  • ATP Binding Cassette Transporter, Subfamily G, Member 8
  • ATP-Binding Cassette Transporters
  • Apolipoproteins E
  • Cholesterol, Dietary
  • Lipoproteins
  • Phytosterols
  • RNA, Messenger
  • Cholesterol