Regio- and stereospecific syntheses and nitric oxide donor properties of (E)-9- and (E)-10-nitrooctadec-9-enoic acids

Org Lett. 2006 May 25;8(11):2305-8. doi: 10.1021/ol060548w.

Abstract

[reaction: see text] Nitrated fatty acids act as endogenous peroxisome proliferator-activated receptor gamma (PPARgamma) ligands and nitric oxide (NO) donors. We describe the first specific preparation of the two regioisomers of nitrooleic acid, (E)-9-nitrooctadec-9-enoic acid (1) and (E)-10-nitrooctadec-9-enoic acid (2), from cis-cyclooctene and monomethyl azelate, respectively. These syntheses rely upon a Henry condensation between a nine-carbon nitro component and a nine-carbon aldehyde. Preliminary chemiluminescence NO detection studies reveal the ability of these nitrated fatty acids to release NO.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Luminescence
  • Molecular Structure
  • Nitric Oxide / chemistry
  • Nitric Oxide / metabolism
  • Nitric Oxide Donors / chemical synthesis*
  • Nitric Oxide Donors / chemistry*
  • Oleic Acids / chemical synthesis*
  • Oleic Acids / chemistry*
  • Stereoisomerism

Substances

  • Nitric Oxide Donors
  • Oleic Acids
  • Nitric Oxide