Biodegradable nanoparticle delivery of a Th2-biased peptide for induction of Th1 immune responses

J Pharm Pharmacol. 2006 Jun;58(6):739-47. doi: 10.1211/jpp.58.6.0004.

Abstract

The type of immune response developed against the hepatitis B virus (HBV) is crucial in determining the outcome of the disease. The protective effects of vaccine-induced antibody responses against subsequent exposure to HBV are well-established. After the establishment of chronic HBV infection, cell-mediated immune response is curative while humoral response is detrimental. A therapeutic vaccine that could switch the type of response could lead to disease resolution. Hepatitis B core antigen (HBcAg)(129-140) has been identified as a Th2-biased peptide in H-2(b) mice when it is administered along with complete Freund's adjuvant (CFA). We formulated HBcAg(129-140) along with monophosphoryl lipid A in poly(D,L-lactic-co-glycolic acid) (PLGA) nanoparticles. Naive mice immunized with the nanoparticle formulation developed a strong Th1-type response while mice immunized with the control formulation of CFA and peptide did not. We then primed mice with CFA and peptide to establish a Th2-type immune response before administering the nanoparticle formulation. Mice receiving the nanoparticle formulation being primed with CFA still developed a strong Th1-type response, while mice that received incomplete Freund's adjuvant and peptide instead of nanoparticles did not. The ability of PLGA nanoparticles to alter the type of immune response elicited by a peptide, even in the context of an ongoing immune response, makes PLGA nanoparticles a strong candidate for the formulation of therapeutic vaccines.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Female
  • Hepatitis B Core Antigens / administration & dosage*
  • Immunization
  • Interferon-gamma / biosynthesis
  • Lactic Acid / administration & dosage
  • Lipid A / administration & dosage
  • Lipid A / analogs & derivatives
  • Lymphocyte Activation
  • Mice
  • Mice, Inbred C57BL
  • Molecular Sequence Data
  • Nanostructures
  • Peptide Fragments / immunology*
  • Polyglycolic Acid / administration & dosage
  • Polylactic Acid-Polyglycolic Acid Copolymer
  • Polymers / administration & dosage
  • T-Lymphocytes / immunology
  • Th1 Cells / immunology*
  • Th2 Cells / immunology

Substances

  • Hepatitis B Core Antigens
  • Lipid A
  • Peptide Fragments
  • Polymers
  • Polylactic Acid-Polyglycolic Acid Copolymer
  • Polyglycolic Acid
  • Lactic Acid
  • Interferon-gamma
  • monophosphoryl lipid A