Ras stimulation of E2F activity and a consequent E2F regulation of integrin alpha6beta4 promote the invasion of breast carcinoma cells

Cancer Res. 2006 Jun 15;66(12):6288-95. doi: 10.1158/0008-5472.CAN-06-0826.

Abstract

Active Ras proteins contribute to breast carcinogenesis and progression. Here, we provide evidence that active H-Ras regulates the expression and activity of the E2F family of transcription factors in SUM-159 breast carcinoma cells. In addition, we show by using a DNA-binding mutant of E2F, as well as expression of specific E2Fs that are transcriptionally active, that the active E2Fs1-3 can mediate the H-Ras-dependent invasion of SUM-159 cells. The inhibitory E2Fs4-5, in contrast, do not influence invasion. One mechanism by which the active E2Fs promote H-Ras-dependent invasion seems to be their ability to increase expression of the beta4 integrin subunit, a component of the alpha6beta4 integrin that is known to enhance carcinoma invasion. Specifically, expression of E2Fs1-3 increased beta4 mRNA, protein, and cell surface expression. The active E2Fs were unable to stimulate invasion in cells that expressed a beta4 short hairpin RNA. This effect of the active E2Fs on beta4 expression does not seem to result from E2F-mediated beta4 transcription because the beta4 promoter lacks known E2F binding motifs. In summary, the data reported here indicate a novel mechanism by which H-Ras can promote the invasion of breast carcinoma cells. This mechanism links active H-Ras, transcriptionally active E2F, and the alpha6beta4 integrin in a common pathway that culminates in enhanced alpha6beta4-dependent invasion.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Breast Neoplasms / genetics
  • Breast Neoplasms / metabolism*
  • Breast Neoplasms / pathology*
  • Cell Adhesion / physiology
  • Cell Line, Tumor
  • Collagen
  • Drug Combinations
  • E2F Transcription Factors / metabolism*
  • Humans
  • Integrin alpha6beta4 / biosynthesis*
  • Integrin alpha6beta4 / genetics
  • Laminin / metabolism
  • Mice
  • NIH 3T3 Cells
  • Neoplasm Invasiveness
  • Proteoglycans
  • RNA, Messenger / biosynthesis
  • RNA, Messenger / genetics
  • Transfection
  • ras Proteins / genetics
  • ras Proteins / metabolism*

Substances

  • Drug Combinations
  • E2F Transcription Factors
  • Integrin alpha6beta4
  • Laminin
  • Proteoglycans
  • RNA, Messenger
  • matrigel
  • Collagen
  • ras Proteins