Cyclooxygenase-independent effects of aspirin on HT-29 human colon cancer cells, revealed by oligonucleotide microarrays

Biotechnol Lett. 2006 Aug;28(16):1263-70. doi: 10.1007/s10529-006-9084-9. Epub 2006 Jul 4.

Abstract

Aspirin and other non-steroidal anti-inflammatory drugs (NSAIDs) inhibit proliferation of human colon cancer cells in vitro. Transmission electron microscope detected morphological features of apoptosis in the aspirin-treated (5 mM, 72 h) HT-29 cells in which cyclooxygenoase-2 is catalytically inactive. We investigated aspirin-induced genome-wide expression changes in HT-29 cells and further studied the time- and concentration-dependent expression changes in 374 apoptosis-related genes, which is the first to show stimulation of genome-wide expression of HT-29 cells by aspirin. The most marked effects of aspirin are on ribosome assembly and rRNA metabolism, which could explain why the quasi-apoptotic morphological changes are not accompanied by a classical DNA ladder. These findings demonstrate that aspirin induces apoptosis in HT-29 cells, bolstering the hypothesis that apoptosis may be a mechanism by which NSAIDs inhibit colon carcinogenesis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Apoptosis
  • Aspirin / pharmacology*
  • Biotechnology / methods
  • Cluster Analysis
  • Colonic Neoplasms / drug therapy*
  • Cyclooxygenase 2 / pharmacology*
  • Genome
  • HT29 Cells
  • Humans
  • Microscopy, Electron
  • Oligonucleotide Array Sequence Analysis / methods*
  • Phylogeny
  • Tetrazolium Salts / pharmacology
  • Thiazoles / pharmacology
  • Time Factors

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Tetrazolium Salts
  • Thiazoles
  • Cyclooxygenase 2
  • thiazolyl blue
  • Aspirin