FGFR4 Arg388 allele is associated with resistance to adjuvant therapy in primary breast cancer

J Clin Oncol. 2006 Aug 10;24(23):3747-55. doi: 10.1200/JCO.2005.04.8587. Epub 2006 Jul 5.

Abstract

Purpose: A recent study presented first evidence that a single nucleotide polymorphism (SNP) at codon 388 of fibroblast growth factor receptor 4 (FGFR4) gene, causing a transmembrane domain missense mutation (Gly388Arg), is associated with disease outcome in node-positive breast cancer. This article addresses the clinical relevance of this SNP, FGFR4 genotype, phenotype, and HER2 regarding patient outcome and influence of adjuvant systemic therapy in a substantial primary breast cancer collective (n = 372; median follow-up, 94.5 months).

Methods: Polymerase chain reaction restriction fragment length polymorphism analysis of germ-line polymorphism was performed in uninvolved lymph nodes; FGFR4 and HER2 expression were assessed immunohistochemically in tissue microarrays.

Results: In 51% of patients, homo- or heterozygous Arg388 allele was present. No correlation existed between FGFR4 genotype and expression or HER2 status. In node-negative patients, FGFR4 genotype was not correlated with disease outcome. In node-positive patients, however, FGFR4 Arg388 was significantly associated with poor disease-free survival (DFS; P = .02) and overall survival (OS; P = .04). Notably, this association seems to be attributable to relatively poor therapy response in Arg388 carriers, reflected in their significantly shorter DFS (P = .02) and OS (P = .045) among patients receiving adjuvant systemic therapy. It is also seen as a significant interaction term in a multivariate proportional hazards model with Arg388 carriers having only about half as much benefit from adjuvant systemic therapy as wild-type carriers.

Conclusion: According to this study, FGFR4 Arg388 genotype is a marker for breast cancer progression in patients with adjuvant systemic therapy, particularly chemotherapy, and thus may indicate therapy resistance.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Alleles
  • Antineoplastic Combined Chemotherapy Protocols / pharmacology*
  • Arginine
  • Biomarkers, Tumor / metabolism*
  • Breast Neoplasms / drug therapy*
  • Breast Neoplasms / genetics*
  • Breast Neoplasms / metabolism
  • Chemotherapy, Adjuvant
  • Disease Progression
  • Drug Resistance, Neoplasm*
  • Female
  • Genetic Markers
  • Genotype
  • Glycine
  • Humans
  • Immunohistochemistry
  • Middle Aged
  • Multivariate Analysis
  • Mutation, Missense
  • Phenotype
  • Polymorphism, Single Nucleotide
  • Predictive Value of Tests
  • Prognosis
  • Proportional Hazards Models
  • Receptor, Fibroblast Growth Factor, Type 4 / genetics*
  • Receptor, Fibroblast Growth Factor, Type 4 / metabolism

Substances

  • Biomarkers, Tumor
  • Genetic Markers
  • Arginine
  • Receptor, Fibroblast Growth Factor, Type 4
  • Glycine