Cell cycle arrest and apoptosis induced by oxaliplatin (L-OHP) on four human cancer cell lines

Anticancer Res. 2006 May-Jun;26(3A):2093-9.

Abstract

Background: The effects of oxaliplatin (L-OHP) on cell cycle and apoptosis were examined.

Materials and methods: The HT29, MCF7, Hela and A549 cell lines were treated and dual parameter flow cytometry BrdU/PI was then performed to monitor cell cycle modifications. Annexin V-FITC and PI probes were used for the detection of apoptosis.

Results: The cells were treated for 3 h followed or not by 24 and 72 h of post-incubation. No changes were observed after 3 h of treatment, while after 24 h of post-incubation, all the cells except A549 were predominantly accumulated in the G2/M-phase; this accumulation was time-dependent. Apoptosis induction was late and moderate and was observed only after 12 h of treatment and 24 h of post-incubation.

Conclusion: L-OHP induced cell cycle arrest and moderate apoptosis; these two activities were time-dependent. These findings warrant further investigation into the potential antitumour activity of L-OHP in MCF7 and Hela cells and in lengthening the infusion duration in order to achieve the acquired cellular modifications.

MeSH terms

  • Antineoplastic Agents / pharmacology*
  • Apoptosis / drug effects*
  • Cell Cycle / drug effects
  • Cell Line, Tumor
  • DNA, Neoplasm / biosynthesis
  • Flow Cytometry
  • HT29 Cells
  • HeLa Cells
  • Humans
  • Organoplatinum Compounds / pharmacology*
  • Oxaliplatin

Substances

  • Antineoplastic Agents
  • DNA, Neoplasm
  • Organoplatinum Compounds
  • Oxaliplatin