Regulation of the Ets-1 transcription factor by sumoylation and ubiquitinylation

Oncogene. 2007 Jan 18;26(3):395-406. doi: 10.1038/sj.onc.1209789. Epub 2006 Jul 24.

Abstract

Sumoylation and ubiquitinylation reversibly regulate the activity of transcription factors through covalent attachment to lysine residues of target proteins. We examined whether the Ets-1 transcription factor is modified by sumoylation and/or ubiquitinylation. Among four potential SUMO motifs in Ets-1, we identified lysines 15 and 227 within the LK(15)YE and IK(227)QE motifs, as being the sumoylation acceptor sites. Using transfection of Ets-1 wildtype (WT) or its sumoylation deficient version (Ets-1 K15R/K227R), as well as WT or mutant proteins of the SUMO pathway, we further demonstrated that the E2 SUMO-conjugating enzyme Ubc9 and a E3 SUMO ligase, PIASy, can enhance Ets-1 sumoylation, while a SUMO protease, SENP1, can desumoylate Ets-1. We also found that Ets-1 is modified by K48-linked polyubiquitinylation independently of the sumoylation acceptor sites and is degraded through the 26S proteasome pathway, while sumoylation of Ets-1 does not affect its stability. Finally, sumoylation of Ets-1 leads to reduced transactivation and we demonstrated that previously identified critical lysine residues in Synergistic Control motifs are the sumoylation acceptor sites of Ets-1. These data show that Ets-1 can be modified by sumoylation and/or ubiquitinylation, with sumoylation repressing transcriptional activity of Ets-1 and having no clear antagonistic action on the ubiquitin-proteasome degradation pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • COS Cells
  • Cell Line
  • Chlorocebus aethiops
  • Dogs
  • Humans
  • Immunoblotting
  • Immunoprecipitation
  • Kidney / metabolism
  • Luciferases / genetics
  • Luciferases / metabolism
  • Protein Processing, Post-Translational*
  • Proto-Oncogene Protein c-ets-1 / genetics
  • Proto-Oncogene Protein c-ets-1 / metabolism*
  • Rabbits
  • SUMO-1 Protein / metabolism*
  • Transcription, Genetic*
  • Ubiquitin / metabolism*
  • Ubiquitin-Conjugating Enzymes / metabolism

Substances

  • Proto-Oncogene Protein c-ets-1
  • SUMO-1 Protein
  • Ubiquitin
  • Luciferases
  • Ubiquitin-Conjugating Enzymes