Prevalence of amiodarone-related hepatotoxicity in 720 Chinese patients with or without baseline liver dysfunction

Clin Cardiol. 2006 Jul;29(7):295-9. doi: 10.1002/clc.4960290705.

Abstract

Background: The prevalence of hepatotoxicity after longterm oral amiodarone therapy in Chinese patients with or without elevated liver enzymes at baseline is unknown.

Hypothesis: Amiodarone may still be safely prescribed for Chinese patients who have baseline liver dysfunction.

Methods: This is a retrospective cross-sectional study. Significant liver dysfunction (SLD) was defined as alanine aminotransferase (ALT) > 2 times upper limit of normal range.

Results: Baseline liver function was checked in 628 of the 720 Chinese patients identified. The mean duration of amiodarone use was 615.9 +/- 703.1 days. Ninety patients (14.3%) had elevated baseline ALT. The prevalence of SLD was 3.7% (confidence interval [CI] 2.1-5.3%) and 4.4% (CI 0.2-8.6%) in patients with normal (n = 538) and elevated (n = 90) baseline ALT, respectively (p = 0.765). Therapy was continued in 42 patients with elevated baseline ALT until final follow-up. Eight of these (19.0%) had elevated ALT upon final follow-up, but the derangement was mild (mean ALT 134.8 +/- 145.9 IU/l, median 76 IU/l). During follow up, 24 patients developed SLD and half of these subsequently withdrew from therapy. The ALT levels at final follow-up had improved over time in both groups, but the mean difference was not significant (255.1 +/- 706.4 vs. 131.0 +/- 207.5 IU/l, p = 0.312).

Conclusion: The prevalence of SLD in Chinese patients taking oral amiodarone with or without elevated baseline ALT was similar (4.4 vs. 3.7%). It seems that amiodarone may be safely prescribed in patients with elevated baseline ALT.

Publication types

  • Multicenter Study

MeSH terms

  • Alanine Transaminase / blood
  • Algorithms
  • Amiodarone / adverse effects*
  • Anti-Arrhythmia Agents / adverse effects*
  • Atrial Fibrillation / drug therapy
  • Atrial Flutter / drug therapy
  • Chemical and Drug Induced Liver Injury / epidemiology*
  • Chemical and Drug Induced Liver Injury / etiology
  • China
  • Cross-Sectional Studies
  • Female
  • Humans
  • Liver / drug effects*
  • Liver Diseases
  • Liver Function Tests
  • Male
  • Prevalence
  • Retrospective Studies
  • Tachycardia / drug therapy

Substances

  • Anti-Arrhythmia Agents
  • Alanine Transaminase
  • Amiodarone