Beta1 integrins: zip codes and signaling relay for blood cells

Curr Opin Cell Biol. 2006 Oct;18(5):482-90. doi: 10.1016/j.ceb.2006.08.007. Epub 2006 Aug 17.

Abstract

At least eight of the twelve known members of the beta1 integrin family are expressed on hematopoietic cells. Among these, the VCAM-1 receptor alpha4beta1 has received most attention as a main factor mediating firm adhesion to the endothelium during blood cell extravasation. Therapeutic trials are ongoing into the use of antibodies and small molecule inhibitors to target this interaction and hence obtain anti-inflammatory effects. However, extravasation is only one possible process that is mediated by beta1 integrins and there is evidence that they also mediate leukocyte retention and positioning in the tissue, lymphocyte activation and possibly migration within the interstitium. Genetic mouse models where integrins are selectively deleted on blood cells have been used to investigate these functions and further studies will be invaluable to critically evaluate therapeutic trials.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / metabolism
  • Anti-Inflammatory Agents / pharmacology
  • Basement Membrane / metabolism
  • Basement Membrane / ultrastructure
  • Blood Cells / drug effects
  • Blood Cells / metabolism*
  • Cell Movement / physiology
  • Endothelium, Vascular / metabolism
  • Endothelium, Vascular / ultrastructure
  • Humans
  • Integrin alpha4beta1 / metabolism*
  • Integrin beta1 / metabolism*
  • Signal Transduction / physiology*

Substances

  • Anti-Inflammatory Agents
  • Integrin alpha4beta1
  • Integrin beta1