Abstract
The neuronal ubiquitin/proteasomal pathway has been implicated in the pathogenesis of Alzheimer's disease (AD). We now show that a component of the pathway, ubiquitin C-terminal hydrolase L1 (Uch-L1), is required for normal synaptic and cognitive function. Transduction of Uch-L1 protein fused to the transduction domain of HIV-transactivator protein (TAT) restores normal enzymatic activity and synaptic function both in hippocampal slices treated with oligomeric Abeta and in the APP/PS1 mouse model of AD. Moreover, intraperitoneal injections with the fusion protein improve the retention of contextual learning in APP/PS1 mice over time. The beneficial effect of the Uch-L1 fusion protein is associated with restoration of normal levels of the PKA-regulatory subunit IIalpha, PKA activity, and CREB phosphorylation.
Publication types
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Research Support, N.I.H., Extramural
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Research Support, Non-U.S. Gov't
MeSH terms
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Alzheimer Disease / enzymology
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Alzheimer Disease / physiopathology*
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Amyloid beta-Protein Precursor / genetics
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Amyloid beta-Protein Precursor / metabolism*
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Animals
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Avoidance Learning
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Cyclic AMP Response Element-Binding Protein / metabolism
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Cyclic AMP-Dependent Protein Kinases / metabolism
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Disease Models, Animal
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Excitatory Postsynaptic Potentials / physiology
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Fear
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Gene Products, tat / genetics
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Gene Products, tat / metabolism
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Hippocampus / cytology
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Hippocampus / metabolism
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Humans
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In Vitro Techniques
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Long-Term Potentiation / physiology
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Membrane Proteins / genetics
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Membrane Proteins / metabolism
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Memory / physiology*
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Mice
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Mice, Inbred C57BL
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Mice, Transgenic
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Presenilin-1
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Recombinant Fusion Proteins / genetics
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Recombinant Fusion Proteins / metabolism*
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Synaptic Transmission / physiology*
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Ubiquitin Thiolesterase / genetics
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Ubiquitin Thiolesterase / metabolism*
Substances
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Amyloid beta-Protein Precursor
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Cyclic AMP Response Element-Binding Protein
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Gene Products, tat
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Membrane Proteins
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PSEN1 protein, human
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Presenilin-1
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Recombinant Fusion Proteins
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UCHL1 protein, human
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Cyclic AMP-Dependent Protein Kinases
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Ubiquitin Thiolesterase
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Uchl1 protein, mouse