Cation binding in Na,K-ATPase, investigated by 205Tl solid-state NMR spectroscopy

Biochemistry. 2006 Sep 5;45(35):10768-76. doi: 10.1021/bi060642k.

Abstract

Cation binding to Na,K-ATPase is characterized in native membranes at room temperature by solid-state NMR spectroscopy using the K(+) congener (205)Tl. It has been demonstrated that the signals from occluded Tl(+) and nonspecifically bound Tl(+) can be detected and distinguished by NMR. Effects of dipole-dipole coupling between (1)H and (205)Tl in the occlusion sites show that the ions are rigidly bound, rather than just occluded. Furthermore, a low chemical shift suggests occlusion site geometries with a relatively small contribution from carboxylate and hydroxyl groups. Nonspecific binding of Tl(+) is characterized by rapid chemical exchange, in agreement with the observed low binding affinity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Binding Sites
  • Cations / chemistry*
  • In Vitro Techniques
  • Kidney / enzymology
  • Kinetics
  • Magnetic Resonance Spectroscopy / methods*
  • Membranes / chemistry*
  • Potassium / chemistry*
  • Protein Binding
  • Salt Gland / enzymology
  • Sharks
  • Sodium-Potassium-Exchanging ATPase / chemistry*
  • Swine

Substances

  • Cations
  • Sodium-Potassium-Exchanging ATPase
  • Potassium