The dynamic pattern of glucocorticoid receptor-mediated transcriptional responses in neuronal PC12 cells

J Neurochem. 2006 Nov;99(4):1282-98. doi: 10.1111/j.1471-4159.2006.04187.x. Epub 2006 Oct 2.

Abstract

The aim of the current study was (i) to examine the overlap in the pattern of glucocorticoid receptor (GR)-mediated transcriptional responses between different neuronal substrates and (ii) to assess the nature of these responses by differentiating between primary and downstream GR-responsive genes. For this purpose, nerve growth factor-differentiated catecholaminergic PC12 cells were used in which endogenous GRs were activated briefly with a high dose of corticosterone followed by gene expression profiling 1 and 3 h afterwards using Affymetrix GeneChips. The results revealed a strikingly similar temporal pattern to that which was reported previously in hippocampus, with only down-regulated genes 1 h after GR activation and the majority of genes up-regulated 3 h after GR activation. Real-time quantatitive PCR of transcripts in cycloheximide-treated cells showed that all five GR-responsive genes selected from the 1-h time point were primary responsive, whereas all four GR-responsive genes selected from the 3-h time point were downstream responsive. At the level of individual genes, the overlap with the previously generated hippocampal data sets was small, illustrating the cell-type specifity of GR-mediated genomic responses. Finally, we identified a number of interesting genes, such as SWI/SNF, synaptosomal-associated protein 25 and certain Rab proteins which may play a role in the effects of glucocorticoids on catecholaminergic neuronal functioning.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain / metabolism*
  • Catecholamines / metabolism
  • Chromosomal Proteins, Non-Histone / genetics
  • Corticosterone / metabolism
  • Corticosterone / pharmacology
  • Cycloheximide / pharmacology
  • Gene Expression Profiling
  • Gene Expression Regulation / drug effects
  • Gene Expression Regulation / genetics*
  • Hippocampus / drug effects
  • Hippocampus / metabolism
  • Nerve Tissue Proteins / biosynthesis*
  • Nerve Tissue Proteins / genetics
  • Neurons / metabolism*
  • PC12 Cells
  • Protein Synthesis Inhibitors / pharmacology
  • Rats
  • Receptors, Glucocorticoid / drug effects
  • Receptors, Glucocorticoid / genetics*
  • Receptors, Glucocorticoid / metabolism
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Synaptosomal-Associated Protein 25 / genetics
  • Time Factors
  • Transcription Factors / genetics
  • Transcriptional Activation / drug effects*
  • Transcriptional Activation / genetics
  • Up-Regulation / drug effects
  • Up-Regulation / genetics
  • rab GTP-Binding Proteins / genetics

Substances

  • Catecholamines
  • Chromosomal Proteins, Non-Histone
  • Nerve Tissue Proteins
  • Protein Synthesis Inhibitors
  • Receptors, Glucocorticoid
  • SWI-SNF-B chromatin-remodeling complex
  • Synaptosomal-Associated Protein 25
  • Transcription Factors
  • Cycloheximide
  • rab GTP-Binding Proteins
  • Corticosterone