Inhibition of L-type but not T-type calcium channel current by a new dihydropyridine derivative, S11568

J Cardiovasc Pharmacol. 1991 Feb;17(2):348-50. doi: 10.1097/00005344-199102000-00024.

Abstract

S11568, (+-)[((amino-2-ethoxy)-2-ethoxy]-methyl)-2-(dichloro-2', 3'-phenyl)-4-ethoxycarbonyl-3-methoxycarbonyl-5-methyl-6-dihydro-1,4-pyr idine HCl, is a new dihydropyridine derivative that is water soluble and relatively insensitive to light. The Ca2+ channel inhibitory activity of S11568 was tested in whole-cell patch clamp recordings from cultured embryonic chick cardiomyocytes in 40 mM Ba2(+)-containing medium that revealed T-type and L-type components of inward current through calcium channels. S11568 inhibited L-type Ca2+ current with an IC50 value near 1 microM but was without effect on the T-type barium current.

MeSH terms

  • Animals
  • Barium / physiology
  • Calcium Channel Blockers / pharmacology*
  • Calcium Channels / drug effects*
  • Chick Embryo
  • Dihydropyridines / pharmacology*
  • Heart / drug effects
  • Heart / embryology

Substances

  • Calcium Channel Blockers
  • Calcium Channels
  • Dihydropyridines
  • S 11568
  • Barium