[Complementary addressed alkylation of 16S rRNA of Escherichia coli by 2',3'-O-[4-N-methyl-N-(2-chloroethyl)-amino]benzylidene derivatives of oligodeoxyribonucleotides. V. Study of the factors affecting selectivity of modification]

Bioorg Khim. 1991 Apr;17(4):470-81.
[Article in Russian]

Abstract

We studied the effect of different factors (reagent concentration, temperature, presence of oligonucleotide-effector (3',5'-diphenazinium derivative of oligodeoxyribonucleotide) stabilizing duplex RNA.reagent) on the selectivity of the site-directed modification of 16S rRNA with 2,3'-O-[4-N-methyl-N-(2-chloroethyl)-amino]-benzylidene derivative of oligonucleotide p(dTTTGCTCCCC)rA (reagent I) under conditions of secondary structure stability. The constant of cooperative binding of the reagent and oligonucleotide-effector with 16s rRNA was determined. The temperature rise from 20 to 40 degrees C brought about a 1.5-fold increase in the relative extent of modification at the target site 771-781. In the presence of oligonucleotide-effector, which is a full complementary copy of the 782-789 fragment of 16S rRNA (reagent concentration is 1 x 10(-6) M), the selectivity of the RNA modification at the target site is doubled and a high level of the modification is retained. When the reagent concentration in the reaction mixture was decreased down to 1 x 10(-7) M, the same level of selectivity was achieved without the oligonucleotide-effector. Under these conditions, however, a drastic (20-fold) drop of the level of the 16S rRNA alkylation was observed.

MeSH terms

  • Alkylation
  • Base Sequence
  • Benzylidene Compounds / chemistry*
  • Escherichia coli / metabolism*
  • Indicators and Reagents
  • Molecular Sequence Data
  • Nitrogen Mustard Compounds / chemistry*
  • Nucleic Acid Conformation
  • Oligodeoxyribonucleotides / chemistry*
  • RNA, Bacterial / chemistry*
  • RNA, Ribosomal, 16S / chemistry*
  • Temperature

Substances

  • Benzylidene Compounds
  • Indicators and Reagents
  • Nitrogen Mustard Compounds
  • Oligodeoxyribonucleotides
  • RNA, Bacterial
  • RNA, Ribosomal, 16S