Comparison of topical dry eye medications for the treatment of keratoconjunctivitis sicca in a botulinum toxin B-induced mouse model

Cornea. 2007 Jan;26(1):84-9. doi: 10.1097/01.ico.0000240079.24583.a1.

Abstract

Purpose: To compare the effects of topical dry eye medications including anti-inflammatory agents and lubricant eyedrops for the treatment of keratoconjunctivitis sicca (KCS) in a botulinum toxin B (BTX-B)-induced mouse model.

Methods: CBA mice were randomized into 10 groups. The first 5 groups received a transconjunctival injection of saline into the lacrimal gland, and the remaining groups were injected with 0.05 mL of 20 mU BTX-B. Each group received treatment with 0.1% fluorometholone (FML), 0.05% cyclosporine A (CsA), a 50:50 combination of FML and CsA, artificial tears, or saline 3 days after injections. Tear production, corneal staining, and blink rate were compared in each of the 10 groups.

Results: Tear production in BTX-B-injected CsA-treated, FML-treated, and combined-treated groups started to return to baseline level within 2 weeks of treatment, whereas those treated with saline or artificial tears still exhibited reduction of lacrimation up to 4 weeks after injection. Topical FML significantly reversed the staining score within 1 week of treatment. The improvement of corneal staining in BTX-B-challenged combined-treated and CsA-treated groups occurred later within 2 weeks after treatment. No significant improvement in corneal staining was observed for the BTX-B-injected mice treated with artificial tears or saline. No significant changes were noted in blink frequency between the control and study groups undergoing the various dry eye therapies.

Conclusion: The therapeutic effects of dry eye medications in a BTX-B-induced mouse model of KCS are similar to the human response.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Topical
  • Animals
  • Blinking
  • Botulinum Toxins / toxicity
  • Botulinum Toxins, Type A
  • Cornea / metabolism
  • Cyclosporine / administration & dosage*
  • Cyclosporine / therapeutic use
  • Disease Models, Animal
  • Drug Therapy, Combination
  • Female
  • Fluorescent Dyes
  • Fluorometholone / administration & dosage*
  • Fluorometholone / therapeutic use
  • Keratoconjunctivitis Sicca / chemically induced
  • Keratoconjunctivitis Sicca / drug therapy*
  • Keratoconjunctivitis Sicca / metabolism
  • Mice
  • Mice, Inbred CBA
  • Ophthalmic Solutions / administration & dosage*
  • Ophthalmic Solutions / therapeutic use
  • Sodium Chloride / administration & dosage
  • Sodium Chloride / therapeutic use
  • Staining and Labeling
  • Tears / metabolism

Substances

  • Fluorescent Dyes
  • Ophthalmic Solutions
  • rimabotulinumtoxinB
  • Sodium Chloride
  • Cyclosporine
  • Botulinum Toxins
  • Botulinum Toxins, Type A
  • Fluorometholone