Boronated DNA-binding compounds as potential agents for boron neutron capture therapy

Mini Rev Med Chem. 2007 Mar;7(3):303-13. doi: 10.2174/138955707780059808.

Abstract

Boron Neutron Capture Therapy (BNCT) is a binary cancer treatment that exploits the short range particles released from a nuclear fission reaction involving the non-radioactive 10B nucleus and low-energy (thermal) neutrons for the destruction of tumour cells. If boronated agents are targeted towards chromosomal DNA, the efficiency of BNCT is greatly enhanced. This article presents a concise review of DNA-binding compounds that have been functionalised with boron.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Review

MeSH terms

  • Alkylating Agents / chemistry
  • Alkylating Agents / therapeutic use
  • Animals
  • Boron Compounds / chemistry*
  • Boron Compounds / therapeutic use
  • Boron Neutron Capture Therapy*
  • DNA / chemistry*
  • Humans
  • Intercalating Agents / chemistry
  • Intercalating Agents / therapeutic use
  • Molecular Structure
  • Neoplasms / radiotherapy*
  • Nucleosides / chemistry

Substances

  • Alkylating Agents
  • Boron Compounds
  • Intercalating Agents
  • Nucleosides
  • DNA