Duloxetine pharmacokinetics are similar in Japanese and Caucasian subjects

Br J Clin Pharmacol. 2007 Mar;63(3):310-4. doi: 10.1111/j.1365-2125.2006.02770.x. Epub 2006 Sep 12.

Abstract

Aims: To compare single- and multiple-dose duloxetine pharmacokinetics between healthy Japanese and Caucasians.

Methods: Twenty-four subjects of each race were given single oral doses of duloxetine (20, 40 and 60 mg) in a randomized, double-blind study. Another 20 subjects of each race received 20, 40 mg or placebo (2 : 2 : 1) twice-daily for 5 days.

Results: Following single doses, the mean duloxetine C(max) and AUC were approximately 20% greater in Japanese. This difference could be explained by the 15% lower average body weight in Japanese. Similar results were observed following multiple dosing.

Conclusion: Duloxetine pharmacokinetics are not meaningfully different between Japanese and Caucasians.

Publication types

  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antidepressive Agents / administration & dosage
  • Antidepressive Agents / pharmacokinetics*
  • Asian People
  • Dose-Response Relationship, Drug
  • Double-Blind Method
  • Duloxetine Hydrochloride
  • Humans
  • Thiophenes / administration & dosage
  • Thiophenes / pharmacokinetics*
  • White People

Substances

  • Antidepressive Agents
  • Thiophenes
  • Duloxetine Hydrochloride