Role of cyclin-dependent kinase 5 in capsaicin-induced cough

Eur J Pharmacol. 2007 Jul 2;566(1-3):181-4. doi: 10.1016/j.ejphar.2007.03.036. Epub 2007 Mar 30.

Abstract

The role of cyclin-dependent kinase 5 (Cdk5) in the capsaicin-induced cough reflex was examined in mice. Pretreatment with inhaled roscovitine, a selective Cdk5 inhibitor, at concentrations of 0.3 to 3 mM inhibited the number of capsaicin-induced coughs in a concentration-dependent manner. Pretreatment with inhaled roscovitine, at a concentration of 3 mM also slightly but significantly inhibited the number of citric acid-induced coughs. The number of capsaicin-induced coughs was significantly reduced when C-fibers were desensitized by the pretreatment with capsaicin. The number of citric acid-induced coughs was slightly but significantly reduced in capsaicin-pretreated mice as compared with that in naive mice. Although the inhalation of roscovitine at a concentration of 3 mM significantly reduced the number of citric acid-induced coughs in naive mice to the level observed in capsaicin-pretreated mice, roscovitine had no effect on the number of citric acid-induced coughs in capsaicin-pretreated mice. These results suggest that Cdk5-dependent factors are involved in C-fiber-mediated cough signaling.

MeSH terms

  • Animals
  • Antitussive Agents / pharmacology*
  • Capsaicin
  • Citric Acid
  • Cough / chemically induced
  • Cough / drug therapy*
  • Cyclin-Dependent Kinase 5 / antagonists & inhibitors*
  • Male
  • Mice
  • Mice, Inbred ICR
  • Protein Kinase Inhibitors / pharmacology*
  • Purines / pharmacology*
  • Roscovitine

Substances

  • Antitussive Agents
  • Protein Kinase Inhibitors
  • Purines
  • Roscovitine
  • Citric Acid
  • Cyclin-Dependent Kinase 5
  • Capsaicin