Expression and possible functions of the cholinergic system in a murine embryonic stem cell line

Life Sci. 2007 May 30;80(24-25):2375-9. doi: 10.1016/j.lfs.2007.03.008. Epub 2007 Mar 19.

Abstract

The expression of a cholinergic system during embryonic development is a widespread phenomenon. However, no precise function could be assigned to it during early pre-neural stages and there are only few studies that document when it precisely starts to be expressed. Here, we examined the expression of cholinergic components in a murine embryonic stem cell line by RT-PCR, histochemistry, and enzyme activity measurements; the acetylcholine (ACh) content was measured by HPLC. We have demonstrated that embryonic stem cells express ACh, acetylcholine receptors, choline acetyltransferase (ChAT), acetyl- and butyryl-cholinesterase (AChE and BChE). Butyryl-cholinesterase (BChE) expression was higher than AChE. The cholinesterase activity was down-regulated by adding specific inhibitors to culture medium. Inhibition of BChE led to a reduction of proliferation. This is the first demonstration that mouse embryonic stem cells express the full molecular equipment of a cholinergic system. Locally produced ACh might function as an intercellular signal, modulating the proliferation of stem cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholine / metabolism
  • Acetylcholinesterase / genetics
  • Acetylcholinesterase / metabolism
  • Animals
  • Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide / pharmacology
  • Butyrylcholinesterase / genetics
  • Butyrylcholinesterase / metabolism
  • Cell Line
  • Cell Proliferation / drug effects
  • Choline O-Acetyltransferase / genetics*
  • Choline O-Acetyltransferase / metabolism
  • Cholinesterase Inhibitors
  • Cholinesterases / genetics*
  • Cholinesterases / metabolism
  • Embryonic Stem Cells / cytology
  • Embryonic Stem Cells / drug effects
  • Embryonic Stem Cells / metabolism*
  • Gene Expression Profiling*
  • Mice
  • Receptors, Cholinergic / genetics*
  • Receptors, Cholinergic / metabolism
  • Reverse Transcriptase Polymerase Chain Reaction
  • Tetraisopropylpyrophosphamide / pharmacology
  • Time Factors

Substances

  • Cholinesterase Inhibitors
  • Receptors, Cholinergic
  • Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide
  • Tetraisopropylpyrophosphamide
  • Choline O-Acetyltransferase
  • Acetylcholinesterase
  • Butyrylcholinesterase
  • Cholinesterases
  • Acetylcholine