p-Coumaric acid inhibits indoleamine 2, 3-dioxygenase expression in murine dendritic cells

Int Immunopharmacol. 2007 Jun;7(6):805-15. doi: 10.1016/j.intimp.2007.01.020. Epub 2007 Feb 27.

Abstract

Indoleamine 2, 3-dioxygenase (IDO), a key enzyme that catalyses the initial and rate-limiting step in the degradation of the tryptophan, is simultaneously expressed in murine dendritic cells and macrophages stimulated with interferon-gamma (IFN-gamma). In the present study, we investigated whether p-Coumaric acid (CA), which is suggested to exhibit antioxidant properties, could suppress the functional expression of IDO in murine bone marrow-derived dendritic cells (BMDCs) stimulated with IFN-gamma. Treatment with CA reduced intracellular expression of IDO mRNA and protein levels in IFN-gamma-activated murine BMDCs in vitro and in CD11c(+)CD8alpha(+) DCs of tumor-draining lymph node (TDLN) of tumor-bearing mice in vivo. Consequently, we obtained evidence that CA suppresses the functional activity of IDO, which catalyses oxidative catabolism of tryptophan, and significantly recovers the IDO-dependent T cell suppression. Activation of the signal transducer and activator of transcription 1 (STAT1) is important to be express IDO in IFN-gamma-stimulated murine BMDCs. To determine whether these inhibitory effects of CA are associated with the alteration of the signal transducer and activator of transcription 1 (STAT1) and IFN-gamma-inducible, dsRNA-activated serine/threonine protein kinase (PKR), BMDCs were pretreated with various concentrations of CA. We found that CA inhibited the activation of STAT1 in response to IFN-gamma. Based on our results, this study may account that CA could inhibit IDO expression by down-regulation of STAT1 activation in IFN-gamma-stimulated murine DCs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Proliferation / drug effects
  • Cells, Cultured
  • Coumaric Acids / pharmacology*
  • Dendritic Cells / drug effects*
  • Dendritic Cells / immunology
  • Immunologic Factors / pharmacology*
  • Indoleamine-Pyrrole 2,3,-Dioxygenase / antagonists & inhibitors*
  • Indoleamine-Pyrrole 2,3,-Dioxygenase / genetics
  • Indoleamine-Pyrrole 2,3,-Dioxygenase / immunology
  • Interferon-gamma / pharmacology
  • Lymph Nodes / cytology
  • Lymph Nodes / immunology
  • Male
  • Melanoma, Experimental / immunology
  • Mice
  • Mice, Inbred BALB C
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • Ovalbumin / immunology
  • Propionates
  • RNA, Messenger / biosynthesis
  • Receptors, Antigen, T-Cell / genetics
  • STAT1 Transcription Factor / immunology
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / immunology

Substances

  • Coumaric Acids
  • Immunologic Factors
  • Indoleamine-Pyrrole 2,3,-Dioxygenase
  • Propionates
  • RNA, Messenger
  • Receptors, Antigen, T-Cell
  • STAT1 Transcription Factor
  • Stat1 protein, mouse
  • Interferon-gamma
  • Ovalbumin
  • p-coumaric acid