Modulation of the K(v)4.3 channel by syntaxin 1A

Biochem Biophys Res Commun. 2007 Jul 6;358(3):789-95. doi: 10.1016/j.bbrc.2007.04.182. Epub 2007 May 4.

Abstract

The SNARE protein syntaxin 1A (Syn1A) is known to inhibit delayed rectifier K(+) channels of the K(v)1 and K(v)2 families with heterogeneous effects on their gating properties. In this study, we explored whether Syn1A could directly modulate K(v)4.3, a rapidly inactivating K(v) channel with important roles in neuroendocrine cells and cardiac myocytes. Immunoprecipitation studies in HEK293 cells coexpressing Syn1A and K(v)4.3 revealed a direct interaction with increased trafficking to the plasma membrane without a change in channel synthesis. Paradoxically, Syn1A inhibited K(v)4.3 current density. In particular, Syn1A produced a left-shift in steady-state inactivation of K(v)4.3 without affecting either voltage dependence of activation or gating kinetics, a pattern distinct from other K(v) channels. Combined with our previous reports, our results further verify the notion that the mechanisms involved in Syn1A-K(v) interactions vary significantly between K(v) channels, thus providing a wide scope for Syn1A modulation of exocytosis and membrane excitability.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line
  • Cell Membrane / metabolism
  • DNA, Complementary / metabolism
  • Electrophysiology
  • Gene Expression Regulation*
  • Humans
  • Immunoprecipitation
  • Kinetics
  • Potassium / chemistry
  • Protein Structure, Tertiary
  • Shal Potassium Channels / chemistry*
  • Subcellular Fractions
  • Syntaxin 1 / chemistry
  • Syntaxin 1 / physiology*
  • Time Factors
  • Transfection

Substances

  • DNA, Complementary
  • Shal Potassium Channels
  • Syntaxin 1
  • Potassium