Dienogest inhibits BrdU uptake with G0/G1 arrest in cultured endometriotic stromal cells

Fertil Steril. 2008 May;89(5 Suppl):1344-7. doi: 10.1016/j.fertnstert.2007.03.042. Epub 2007 May 23.

Abstract

Objective: To investigate the effect of dienogest on the proliferation of endometriotic stromal cells.

Design: Comparative and laboratory study.

Setting: University of Tokyo Hospital.

Patient(s): Endometriotic stromal cells were isolated and cultured from ovarian endometriomas of patients undergoing surgery.

Intervention(s): Dienogest was added to the cultured endometriotic stromal cells.

Main outcome measure(s): 5-Bromo-2'-deoxyuridine (BrdU) incorporation into DNA of the endometriotic stromal cells was measured by ELISA. Cell cycle analysis of the cultured endometriotic stromal cells was performed by flow cytometry.

Result(s): Dienogest at concentration of 10(-7) M and 10(-6) M significantly inhibited BrdU incorporation into DNA at 24 and 48 hours. Dienogest significantly increased the cells in G0/G1 phase and reduced the cells in S phase and G2/M phase in 24 and 48 hours.

Conclusion(s): The present study indicates that dienogest can inhibit the proliferation of the endometriotic stromal cells with G0/G1 arrest, suggesting a possible direct effect of dienogest in the treatment of endometriosis.

MeSH terms

  • Adult
  • Bromodeoxyuridine / pharmacokinetics*
  • Cell Cycle / drug effects
  • Cell Proliferation / drug effects*
  • Cells, Cultured
  • Contraceptives, Oral / pharmacology
  • DNA / metabolism
  • Drug Evaluation, Preclinical
  • Endometriosis / metabolism
  • Endometriosis / pathology*
  • Female
  • G1 Phase / drug effects*
  • Humans
  • Nandrolone / analogs & derivatives*
  • Nandrolone / pharmacology
  • Ovarian Diseases / metabolism
  • Ovarian Diseases / pathology*
  • Resting Phase, Cell Cycle / drug effects*
  • Stromal Cells / metabolism
  • Stromal Cells / pathology*

Substances

  • Contraceptives, Oral
  • dienogest
  • Nandrolone
  • DNA
  • Bromodeoxyuridine