An outwardly rectifying anionic background current in atrial myocytes from the human heart

Biochem Biophys Res Commun. 2007 Aug 3;359(3):765-70. doi: 10.1016/j.bbrc.2007.05.177. Epub 2007 Jun 4.

Abstract

This report describes a hitherto unreported anionic background current from human atrial cardiomyocytes. Under whole-cell patch-clamp with anion-selective conditions, an outwardly rectifying anion current (I(ANION)) was observed, which was larger with iodide than nitrate, and with nitrate than chloride as charge carrier. In contrast with a previously identified background anionic current from small mammal cardiomyocytes, I(ANION) was not augmented by the pyrethroid tefluthrin (10 microM); neither was it inhibited by hyperosmolar external solution nor by DIDS (200 microM); thus I(ANION) was not due to basal activity of volume-sensitive anion channels. I(ANION) was partially inhibited by the Cl(-) channel blockers NPPB (50 microM) and Gly H-101 (30 microM). Incorporation of I(ANION) into a human atrial action potential (AP) simulation led to depression of the AP plateau, accompanied by alterations to plateau inward calcium current, and to AP shortening at 50% but not 90% of complete repolarization, demonstrating that I(ANION) can influence the human atrial AP profile.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Anions / metabolism
  • Electric Conductivity
  • Female
  • Heart Atria / cytology*
  • Humans
  • Male
  • Muscle Cells / metabolism*
  • Patch-Clamp Techniques

Substances

  • Anions